TDR Targets

Basic information

Technical information

Name: Unnamed compound
MW: 413.511 | Formula: C26H27N3O2
H donors: 1 H acceptors: 2 LogP: 4.19 Rotable bonds: 8
Rule of 5 violations (Lipinski): 1
SMILES: O=C(C1CCCN(C1)C/C=C/c1ccccc1)Nc1ccccc1Oc1cccnc1
InChi: 1S/C26H27N3O2/c30-26(28-24-14-4-5-15-25(24)31-23-13-6-16-27-19-23)22-12-8-18-29(20-22)17-7-11-21-9-2-1-3-10-21/h1-7,9-11,13-16,19,22H,8,12,17-18,20H2,(H,28,30)/b11-7+
InChiKey: YOKBPLZKZAGVRJ-YRNVUSSQSA-N

Network

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Target Layer

Model Organisms

Species	Viewmode
Arabidopsis thaliana
Caenorhabditis elegans
Dictyostelium discoideum
Drosophila melanogaster
Escherichia coli
Homo sapiens
Mus musculus
Oryza sativa
Saccharomyces cerevisiae
Schmidtea mediterranea
Other organisms

TDR Pathogens:

Species	Viewmode
Brugia malayi
Chlamydia trachomatis
Echinococcus granulosus
Entamoeba histolytica
Echinococcus multilocularis
Giardia lamblia
Leishmania major
Loa Loa (eye worm)
Mycobacterium leprae
Mycobacterium tuberculosis
Mycobacterium ulcerans
Onchocerca volvulus
Plasmodium falciparum
Plasmodium vivax
Schistosoma mansoni
Trypanosoma brucei
Trypanosoma cruzi
Toxoplasma gondii
Treponema pallidum
Trichomonas vaginalis
Wolbachia endosymbiont of Brugia malayi

Other Pathogens:

Species	Viewmode
Babesia bovis
Candida albicans
Cryptosporidium hominis
Cryptosporidium parvum
Leishmania braziliensis
Leishmania donovani
Leishmania infantum
Leishmania mexicana
Neospora caninum
Plasmodium berghei
Plasmodium knowlesi
Plasmodium yoelii
Schistosoma japonicum
Trypanosoma brucei gambiense
Trypanosoma congolense
Theileria parva

Compound Layer

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Clustering layers

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Synonyms

No synonyms found for this compound

Targets

Known targets for this compound

Species	Target name	Source	Bibliographic reference
Homo sapiens	ATPase family, AAA domain containing 5	Starlite/ChEMBL	No references
Homo sapiens	glucagon-like peptide 1 receptor	Starlite/ChEMBL	No references

Predicted pathogen targets for this compound

By orthology

Species	Potential target	Known druggable target/s	Ortholog Group
Echinococcus multilocularis	atpase aaa+ type core atpase aaa type core	Get druggable targets OG5_139225	All targets in OG5_139225

By sequence similarity to non orthologous known druggable targets

Species	Potential target	Known druggable target	Length	Alignment span	Identity
Loa Loa (eye worm)	pigment dispersing factor receptor c	glucagon-like peptide 1 receptor	463 aa	388 aa	25.8 %

Ranking Plot

Putative Targets List

Species	Potential target	Raw	Global	Species
Echinococcus multilocularis	expressed conserved protein	0.0095	0.0259	0.0253
Mycobacterium tuberculosis	Putative acetyl hydrolase MbtJ	0.0051	0.0113	0.1525
Loa Loa (eye worm)	hypothetical protein	0.0101	0.028	0.0277
Mycobacterium ulcerans	esterase/lipase	0.0051	0.0113	0.1235
Mycobacterium tuberculosis	Probable hydrolase	0.0037	0.0068	0.0913
Schistosoma mansoni	hypothetical protein	0.0042	0.0082	0.0076
Onchocerca volvulus		0.0037	0.0068	0.4912
Echinococcus multilocularis	protein dispatched 1	0.0049	0.0108	0.0101
Echinococcus multilocularis	Niemann Pick C1 protein	0.0144	0.0424	0.0418
Mycobacterium tuberculosis	Probable lipase LipH	0.0051	0.0113	0.1525
Trichomonas vaginalis	fructose-bisphosphate aldolase, putative	0.0299	0.0943	1
Mycobacterium tuberculosis	Probable non lipolytic carboxylesterase NlhH	0.0051	0.0113	0.1525
Loa Loa (eye worm)	hypothetical protein	0.0043	0.0087	0.0084
Trichomonas vaginalis	Esterase, putative	0.0051	0.0113	0.1123
Brugia malayi	AMP-binding enzyme family protein	0.0024	0.0024	0.0197
Mycobacterium tuberculosis	Probable lipase/esterase LipN	0.0051	0.0113	0.1525
Mycobacterium ulcerans	lipase LipH	0.0051	0.0113	0.1235
Loa Loa (eye worm)	exodeoxyribonuclease III family protein	0.0019	0.0008	0.0005
Mycobacterium ulcerans	lipase LipU	0.0051	0.0113	0.1235
Mycobacterium tuberculosis	Conserved protein	0.0037	0.0068	0.0913
Mycobacterium leprae	conserved hypothetical protein	0.0037	0.0068	0.1074
Schistosoma mansoni	hormone-sensitive lipase (S09 family)	0.3004	1	1
Mycobacterium ulcerans	carboxylesterase LipQ	0.0051	0.0113	0.1235
Trichomonas vaginalis	fructose-bisphosphate aldolase, putative	0.0299	0.0943	1
Mycobacterium ulcerans	hypothetical protein	0.0024	0.0024	0.0231
Trichomonas vaginalis	penicillin-binding protein, putative	0.0037	0.0068	0.0638
Schistosoma mansoni	hypothetical protein	0.0037	0.0066	0.0059
Schistosoma mansoni	ap endonuclease	0.0019	0.0008	0.0002
Schistosoma mansoni	ap endonuclease	0.0019	0.0008	0.0002
Mycobacterium ulcerans	esterase LipO	0.0051	0.0113	0.1235
Mycobacterium tuberculosis	Probable esterase LipO	0.0051	0.0113	0.1525
Entamoeba histolytica	acyl-CoA synthetase, putative	0.0024	0.0024	0.017
Loa Loa (eye worm)	glutaminase 2	0.0283	0.0891	0.0888
Trypanosoma brucei	Isoprenylcysteine alpha-carbonyl methylesterase, putative	0.0051	0.0113	1
Echinococcus granulosus	Niemann Pick C1 protein	0.0144	0.0424	0.0418
Entamoeba histolytica	acyl-coA synthetase, putative	0.0024	0.0024	0.017
Schistosoma mansoni	hypothetical protein	0.0042	0.0082	0.0076
Loa Loa (eye worm)	hypothetical protein	0.0037	0.0068	0.0064
Loa Loa (eye worm)	abnormal chemotaxis protein 14	0.0043	0.0087	0.0084
Toxoplasma gondii	alpha/beta hydrolase fold domain-containing protein	0.0051	0.0113	1
Mycobacterium tuberculosis	Conserved protein	0.0037	0.0068	0.0913
Mycobacterium tuberculosis	Probable chain -fatty-acid-CoA ligase FadD13 (fatty-acyl-CoA synthetase)	0.0024	0.0024	0.0322
Toxoplasma gondii	ABC1 family protein	0.0037	0.0068	0.5682
Leishmania major	hypothetical protein, conserved	0.0037	0.0068	0.5682
Loa Loa (eye worm)	hypothetical protein	0.0024	0.0024	0.0021
Leishmania major	4-coumarate:coa ligase-like protein	0.0024	0.0024	0.1513
Echinococcus granulosus	beta LACTamase domain containing family member	0.0037	0.0068	0.0061
Brugia malayi	Niemann-Pick C1 protein precursor	0.0101	0.028	0.3088
Mycobacterium tuberculosis	Possible lipase LipU	0.0051	0.0113	0.1525
Trichomonas vaginalis	fructose-bisphosphate aldolase, putative	0.0299	0.0943	1
Mycobacterium ulcerans	exodeoxyribonuclease III protein XthA	0.0019	0.0008	0.0052
Trichomonas vaginalis	fructose-bisphosphate aldolase, putative	0.0299	0.0943	1
Mycobacterium tuberculosis	Probable esterase LipM	0.0051	0.0113	0.1525
Echinococcus multilocularis	Basic leucine zipper (bZIP) transcription	0.0037	0.0066	0.0059
Brugia malayi	Corticotropin releasing factor receptor 2 precursor, putative	0.006	0.0144	0.1557
Echinococcus multilocularis	sterol regulatory element binding protein	0.0043	0.0087	0.0081
Echinococcus granulosus	DNA apurinic or apyrimidinic site lyase	0.0019	0.0008	0.0002
Mycobacterium ulcerans	esterase LipW	0.0051	0.0113	0.1235
Trypanosoma cruzi	hypothetical protein, conserved	0.0037	0.0068	0.5682
Echinococcus multilocularis	DNA (apurinic or apyrimidinic site) lyase	0.0019	0.0008	0.0002
Loa Loa (eye worm)	beta-lactamase	0.0037	0.0068	0.0064
Schistosoma mansoni	niemann-pick C1 (NPC1)	0.0102	0.0285	0.0279
Entamoeba histolytica	hypothetical protein	0.0037	0.0066	0.0619
Trypanosoma cruzi	hypothetical protein, conserved	0.0037	0.0068	0.5682
Trypanosoma brucei	hypothetical protein, conserved	0.0037	0.0068	0.5682
Trypanosoma cruzi	Isoprenylcysteine alpha-carbonyl methylesterase, putative	0.0051	0.0113	1
Trypanosoma cruzi	serine peptidase, Clan SC, Family S9D	0.0051	0.0113	1
Mycobacterium tuberculosis	Probable fatty-acid-CoA ligase FadD2 (fatty-acid-CoA synthetase) (fatty-acid-CoA synthase)	0.0024	0.0024	0.0322
Mycobacterium ulcerans	hypothetical protein	0.0051	0.0113	0.1235
Mycobacterium tuberculosis	Probable carboxylesterase LipQ	0.0051	0.0113	0.1525
Trichomonas vaginalis	conserved hypothetical protein	0.0051	0.0113	0.1123
Mycobacterium leprae	Probable fructose bisphosphate aldolase Fba	0.0146	0.0431	1
Plasmodium falciparum	AP endonuclease (DNA-[apurinic or apyrimidinic site] lyase), putative	0.0019	0.0008	1
Mycobacterium tuberculosis	Probable exodeoxyribonuclease III protein XthA (exonuclease III) (EXO III) (AP endonuclease VI)	0.0019	0.0008	0.0107
Loa Loa (eye worm)	glutaminase	0.0283	0.0891	0.0888
Brugia malayi	exodeoxyribonuclease III family protein	0.0019	0.0008	0.0017
Entamoeba histolytica	acyl-CoA synthetase, putative	0.0024	0.0024	0.017
Treponema pallidum	N-acetylphosphinothricin-tripetide-deacetylase	0.0051	0.0113	0.1123
Schistosoma mansoni	hypothetical protein	0.0041	0.008	0.0074
Loa Loa (eye worm)	hypothetical protein	0.0024	0.0024	0.0021
Brugia malayi	CHE-14 protein	0.0043	0.0087	0.0914
Loa Loa (eye worm)	pigment dispersing factor receptor c	0.006	0.0144	0.0141
Brugia malayi	beta-lactamase family protein	0.0037	0.0068	0.0692
Mycobacterium tuberculosis	Probable lipase LipE	0.0037	0.0068	0.0913
Plasmodium vivax	hypothetical protein, conserved	0.0037	0.0068	1
Mycobacterium tuberculosis	Possible esterase LipW	0.0051	0.0113	0.1525
Mycobacterium ulcerans	acyl-CoA synthetase	0.0024	0.0024	0.0231
Loa Loa (eye worm)	hypothetical protein	0.3004	1	1
Entamoeba histolytica	fructose-1,6-bisphosphate aldolase, putative	0.0299	0.0943	1
Giardia lamblia	Fructose-bisphosphate aldolase	0.0299	0.0943	1
Leishmania major	hypothetical protein, conserved	0.0051	0.0113	1
Entamoeba histolytica	hypothetical protein	0.0037	0.0066	0.0619
Echinococcus granulosus	Protein patched homolog 1	0.0043	0.0087	0.0081
Echinococcus granulosus	Niemann Pick C1 protein	0.0101	0.028	0.0273
Mycobacterium ulcerans	fructose-bisphosphate aldolase	0.0146	0.0431	0.4821
Mycobacterium ulcerans	long-chain fatty-acid CoA ligase	0.0024	0.0024	0.0231
Schistosoma mansoni	hormone-sensitive lipase (S09 family)	0.3004	1	1
Brugia malayi	beta-lactamase	0.0037	0.0068	0.0692
Entamoeba histolytica	Niemann-Pick C1 protein, putative	0.0101	0.028	0.2906
Loa Loa (eye worm)	hypothetical protein	0.0037	0.0068	0.0064
Schistosoma mansoni	hypothetical protein	0.0042	0.0082	0.0076
Brugia malayi	Calcitonin receptor-like protein seb-1	0.006	0.0144	0.1557
Trichomonas vaginalis	penicillin-binding protein, putative	0.0037	0.0068	0.0638
Plasmodium vivax	AP endonuclease (DNA-[apurinic or apyrimidinic site] lyase), putative	0.0019	0.0008	0.0719
Echinococcus multilocularis	beta LACTamase domain containing family member	0.0037	0.0068	0.0061
Mycobacterium ulcerans	lipase LipI	0.0051	0.0113	0.1235
Trichomonas vaginalis	D-aminoacylase, putative	0.0037	0.0068	0.0638
Mycobacterium tuberculosis	Probable esterase/lipase LipF	0.0051	0.0113	0.1525
Mycobacterium ulcerans	hypothetical protein	0.0037	0.0068	0.0724
Entamoeba histolytica	hypothetical protein	0.0037	0.0066	0.0619
Mycobacterium tuberculosis	Probable esterase/lipase LipP	0.0037	0.0068	0.0913
Loa Loa (eye worm)	hypothetical protein	0.006	0.0144	0.0141
Loa Loa (eye worm)	hypothetical protein	0.0037	0.0068	0.0064
Mycobacterium tuberculosis	Possible penicillin-binding protein	0.0238	0.0741	1
Mycobacterium tuberculosis	Probable fructose-bisphosphate aldolase Fba	0.0146	0.0431	0.5823
Mycobacterium tuberculosis	Possible conserved lipoprotein LpqK	0.0037	0.0068	0.0913
Toxoplasma gondii	alpha/beta hydrolase fold domain-containing protein	0.0051	0.0113	1
Mycobacterium leprae	Possible lipase LipU	0.0051	0.0113	0.2187
Loa Loa (eye worm)	hypothetical protein	0.0019	0.0006	0.0003
Mycobacterium ulcerans	lipase/esterase LipN	0.0051	0.0113	0.1235
Trichomonas vaginalis	D-aminoacylase, putative	0.0037	0.0068	0.0638
Trichomonas vaginalis	fructose-bisphosphate aldolase, putative	0.0299	0.0943	1
Trypanosoma cruzi	Isoprenylcysteine alpha-carbonyl methylesterase, putative	0.0051	0.0113	1
Trichomonas vaginalis	glutaminase, putative	0.0283	0.0891	0.9446
Echinococcus granulosus	expressed conserved protein	0.0095	0.0259	0.0253
Mycobacterium ulcerans	acyl-CoA synthetase	0.0024	0.0024	0.0231
Mycobacterium ulcerans	membrane-bound esterase LipM	0.0051	0.0113	0.1235
Schistosoma mansoni	patched 1	0.0043	0.0087	0.0081
Schistosoma mansoni	hypothetical protein	0.0042	0.0082	0.0076
Mycobacterium tuberculosis	Probable esterase LipC	0.0051	0.0113	0.1525
Wolbachia endosymbiont of Brugia malayi	exonuclease III	0.0019	0.0008	0.5
Echinococcus multilocularis	atpase aaa+ type core atpase aaa type core	0.0979	0.3221	0.3216
Mycobacterium ulcerans	lipase LipU	0.0051	0.0113	0.1235
Mycobacterium tuberculosis	Probable lipase LipD	0.0037	0.0068	0.0913
Mycobacterium tuberculosis	Fatty-acid-AMP ligase FadD30 (fatty-acid-AMP synthetase) (fatty-acid-AMP synthase)	0.0018	0.0003	0.0045
Echinococcus granulosus	sterol regulatory element binding protein	0.0043	0.0087	0.0081
Schistosoma mansoni	hormone-sensitive lipase (S09 family)	0.3004	1	1
Loa Loa (eye worm)	hypothetical protein	0.0053	0.012	0.0117
Brugia malayi	AMP-binding enzyme family protein	0.0024	0.0024	0.0197
Mycobacterium leprae	Probable lipase LipE	0.0037	0.0068	0.1074
Echinococcus multilocularis	hormone sensitive lipase	0.3004	1	1
Mycobacterium ulcerans	acetyl hydrolase MbtJ	0.0051	0.0113	0.1235
Loa Loa (eye worm)	latrophilin receptor protein 2	0.0019	0.0006	0.0003
Brugia malayi	glutaminase DH11.1	0.0283	0.0891	1
Trypanosoma cruzi	Alpha/beta hydrolase domain-containing protein	0.0051	0.0113	1
Schistosoma mansoni	family S12 unassigned peptidase (S12 family)	0.0037	0.0068	0.0061
Trichomonas vaginalis	D-aminoacylase, putative	0.0037	0.0068	0.0638
Trichomonas vaginalis	esterase, putative	0.0037	0.0068	0.0638
Brugia malayi	beta-lactamase family protein	0.0037	0.0068	0.0692
Trichomonas vaginalis	Esterase, putative	0.0051	0.0113	0.1123
Loa Loa (eye worm)	hypothetical protein	0.0037	0.0068	0.0064
Mycobacterium ulcerans	fusion of enoyl-CoA hydratase, EchA21 and lipase, LipE	0.0037	0.0068	0.0724
Schistosoma mansoni	family S12 unassigned peptidase (S12 family)	0.0037	0.0068	0.0061
Mycobacterium ulcerans	beta-lactamase	0.0037	0.0068	0.0724
Schistosoma mansoni	transcription factor LCR-F1	0.0037	0.0066	0.0059
Mycobacterium ulcerans	esterase LipC	0.0051	0.0113	0.1235
Onchocerca volvulus		0.0037	0.0068	0.4912
Onchocerca volvulus		0.0051	0.0113	1
Mycobacterium ulcerans	esterase/lipase LipP	0.0037	0.0068	0.0724
Chlamydia trachomatis	acylglycerophosphoethanolamine acyltransferase	0.0018	0.0003	0.5
Schistosoma mansoni	glutaminase	0.0283	0.0891	0.0886
Trichomonas vaginalis	fructose-bisphosphate aldolase, putative	0.0299	0.0943	1
Mycobacterium tuberculosis	Probable acetyl-hydrolase/esterase LipR	0.0051	0.0113	0.1525
Echinococcus granulosus	Basic leucine zipper bZIP transcription	0.0037	0.0066	0.0059
Leishmania major	4-coumarate:coa ligase-like protein	0.0024	0.0024	0.1513
Mycobacterium tuberculosis	Probable conserved lipoprotein	0.0037	0.0068	0.0913
Leishmania major	4-coumarate:coa ligase-like protein	0.0024	0.0024	0.1513
Entamoeba histolytica	hypothetical protein	0.0037	0.0066	0.0619
Brugia malayi	latrophilin 2 splice variant baaae	0.0041	0.008	0.0836
Brugia malayi	aryl-acylamidase	0.0051	0.0113	0.1204
Loa Loa (eye worm)	hypothetical protein	0.0041	0.008	0.0077
Loa Loa (eye worm)	hypothetical protein	0.0037	0.0068	0.0064
Trichomonas vaginalis	conserved hypothetical protein	0.0043	0.0087	0.0849
Mycobacterium ulcerans	long-chain-fatty-acid-CoA ligase	0.0024	0.0024	0.0231
Brugia malayi	hypothetical protein	0.0037	0.0066	0.0671
Leishmania major	ecotin, putative	0.0051	0.0113	1
Mycobacterium ulcerans	acyl-CoA synthetase	0.0024	0.0024	0.0231
Mycobacterium ulcerans	lipase LipD	0.0037	0.0068	0.0724
Mycobacterium tuberculosis	Conserved protein	0.0037	0.0068	0.0913
Entamoeba histolytica	fructose-1,6-bisphosphate aldolase, putative	0.0299	0.0943	1
Treponema pallidum	fructose-bisphosphate aldolase	0.0299	0.0943	1
Loa Loa (eye worm)	hypothetical protein	0.0024	0.0024	0.0021
Mycobacterium ulcerans	fatty-acid-CoA ligase	0.0024	0.0024	0.0231
Onchocerca volvulus		0.0037	0.0068	0.4912
Schistosoma mansoni	family S9 non-peptidase homologue (S09 family)	0.0051	0.0113	0.0107
Trichomonas vaginalis	Esterase, putative	0.0051	0.0113	0.1123
Loa Loa (eye worm)	aryl-acylamidase	0.0051	0.0113	0.011
Brugia malayi	Hypothetical 52.5 kDa protein ZK945.1 in chromosome II, putative	0.0037	0.0068	0.0692
Trichomonas vaginalis	fructose-bisphosphate aldolase, putative	0.0299	0.0943	1
Brugia malayi	AMP-binding enzyme family protein	0.0024	0.0024	0.0197
Loa Loa (eye worm)	beta-LACTamase domain containing family member	0.0037	0.0068	0.0064
Echinococcus multilocularis	Niemann Pick C1 protein	0.0101	0.028	0.0273
Loa Loa (eye worm)	ammd protein	0.0051	0.0113	0.011
Mycobacterium ulcerans	long-chain-fatty-acid--CoA ligase	0.0024	0.0024	0.0231
Echinococcus multilocularis	protein patched	0.0043	0.0087	0.0081
Mycobacterium ulcerans	glutaminase	0.0283	0.0891	1
Trichomonas vaginalis	fructose-bisphosphate aldolase, putative	0.0299	0.0943	1
Mycobacterium tuberculosis	Probable esterase LipL	0.0037	0.0068	0.0913
Loa Loa (eye worm)	hypothetical protein	0.0037	0.0068	0.0064

Activities

Activity type	Activity value	Assay description	Source	Reference
Potency (functional)	5.2213 uM	PUBCHEM_BIOASSAY: Primary qHTS for delayed death inhibitors of the malarial parasite plastid, 48 hour incubation. (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID488752, AID488774, AID504848, AID504850]	ChEMBL.	No reference
Potency (functional)	6.5104 uM	PUBCHEM_BIOASSAY: qHTS screen for small molecules that inhibit ELG1-dependent DNA repair in human embryonic kidney (HEK293T) cells expressing luciferase-tagged ELG1. (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID493107, AID493125]	ChEMBL.	No reference
Potency (functional)	8.9125 uM	PubChem BioAssay. qHTS of GLP-1 Receptor Inverse Agonists (Inhibition Mode). (Class of assay: confirmatory)	ChEMBL.	No reference
Potency (functional)	12.5893 uM	PUBCHEM_BIOASSAY: qHTS for Inhibitors of TGF-b: Cytotox Counterscreen. (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID588855, AID588860]	ChEMBL.	No reference
Potency (functional)	18.526 uM	PUBCHEM_BIOASSAY: Primary qHTS for delayed death inhibitors of the malarial parasite plastid, 96 hour incubation. (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID488745, AID488752, AID488774, AID504848, AID504850]	ChEMBL.	No reference
Potency (functional)	= 39.8107 um	PUBCHEM_BIOASSAY: qHTS Assay for Inhibitors of DNA Polymerase Beta. (Class of assay: confirmatory)	ChEMBL.	No reference

Phenotypes

Whole-cell/tissue/organism interactions

Species name	Source	Reference	Is orphan
Plasmodium falciparum	ChEMBL23
Homo sapiens	ChEMBL23

Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.

Annotated phenotypes:

We have no manually annotated phenotypes for this drug. What does this mean? / Care to help?

In TDR Targets, information about phenotypes that are caused by drugs, or by genetic manipulation of cells (e.g. gene knockouts or knockdowns) is manually curated from the literature. These descriptions help to describe the potential of the target for drug development. If no information is available for this gene or if the information is incomplete, this may mean that i) the papers containing this information either appeared after the curation effort for this organism was carried out or they were inadvertently missed by curators; or that ii) the curation effort for this organism has not yet started.

In any case, if you have information about papers containing relevant validation data for this target, please log in using your TDR Targets username and password and send them to us using the corresponding form in this page (only visible to registered users) or contact us.

External resources for this compound

ChEMBL: CHEMBL1415240

Bibliographic References

No literature references available for this target.

If you have references for this compound, please enter them in a user comment (below) or Contact us.

Detailed information for compound 1308207