Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Wolbachia endosymbiont of Brugia malayi | exonuclease III | 0.0018 | 0.0532 | 0.5 |
Leishmania major | eukaryotic translation initiation factor-like | 0.0112 | 0.4691 | 1 |
Trichomonas vaginalis | set domain proteins, putative | 0.0233 | 1 | 1 |
Echinococcus multilocularis | histone lysine N methyltransferase SETMAR | 0.003 | 0.1038 | 0.138 |
Trichomonas vaginalis | conserved hypothetical protein | 0.0013 | 0.0311 | 0.0311 |
Treponema pallidum | exodeoxyribonuclease (exoA) | 0.0018 | 0.0532 | 0.5 |
Entamoeba histolytica | exodeoxyribonuclease III, putative | 0.0018 | 0.0532 | 0.0505 |
Brugia malayi | latrophilin 2 splice variant baaae | 0.0035 | 0.1252 | 0.1285 |
Mycobacterium tuberculosis | Probable exodeoxyribonuclease III protein XthA (exonuclease III) (EXO III) (AP endonuclease VI) | 0.0018 | 0.0532 | 0.5 |
Echinococcus multilocularis | geminin | 0.0166 | 0.7054 | 1 |
Echinococcus granulosus | diuretic hormone 44 receptor GPRdih2 | 0.0016 | 0.0428 | 0.0506 |
Schistosoma mansoni | hypothetical protein | 0.0166 | 0.7054 | 1 |
Loa Loa (eye worm) | hypothetical protein | 0.0035 | 0.1252 | 0.128 |
Loa Loa (eye worm) | eukaryotic translation initiation factor 4E type 3 | 0.0013 | 0.0311 | 0.0187 |
Brugia malayi | Latrophilin receptor protein 2 | 0.0016 | 0.0428 | 0.0328 |
Echinococcus granulosus | cpg binding protein | 0.003 | 0.1032 | 0.1372 |
Trichomonas vaginalis | eukaryotic translation initiation factor 4E type, putative | 0.0013 | 0.0311 | 0.0311 |
Loa Loa (eye worm) | eukaryotic translation initiation factor 4E-1 | 0.0013 | 0.0311 | 0.0187 |
Trichomonas vaginalis | eukaryotic translation initiation factor 4E type, putative | 0.0013 | 0.0311 | 0.0311 |
Trichomonas vaginalis | eukaryotic translation initiation factor 4E, putative | 0.0013 | 0.0311 | 0.0311 |
Echinococcus granulosus | GPCR family 2 | 0.0016 | 0.0428 | 0.0506 |
Schistosoma mansoni | histone-lysine n-methyltransferase suv9 | 0.003 | 0.1038 | 0.138 |
Schistosoma mansoni | hypothetical protein | 0.0011 | 0.021 | 0.0193 |
Echinococcus multilocularis | histone lysine methyltransferase setb histone lysine methyltransferase eggless | 0.003 | 0.1038 | 0.138 |
Trichomonas vaginalis | eukaryotic translation initiation factor 4E, putative | 0.0013 | 0.0311 | 0.0311 |
Brugia malayi | Eukaryotic translation initiation factor 4E type 3, putative | 0.0013 | 0.0311 | 0.0192 |
Brugia malayi | eukaryotic translation initiation factor 4E-1 | 0.0013 | 0.0311 | 0.0192 |
Echinococcus multilocularis | GPCR, family 2 | 0.0016 | 0.0428 | 0.0506 |
Onchocerca volvulus | 0.003 | 0.1038 | 0.075 | |
Leishmania major | eukaryotic translation initiation factor eIF-4E, putative | 0.0112 | 0.4691 | 1 |
Loa Loa (eye worm) | hypothetical protein | 0.0025 | 0.0814 | 0.0771 |
Schistosoma mansoni | ap endonuclease | 0.0018 | 0.0532 | 0.0656 |
Schistosoma mansoni | cpg binding protein | 0.003 | 0.1032 | 0.1372 |
Brugia malayi | GTP-binding regulatory protein Gs alpha-S chain, putative | 0.0045 | 0.1706 | 0.1812 |
Loa Loa (eye worm) | latrophilin receptor protein 2 | 0.0016 | 0.0428 | 0.0323 |
Schistosoma mansoni | mixed-lineage leukemia protein mll | 0.0061 | 0.2403 | 0.3336 |
Trypanosoma cruzi | Eukaryotic translation initiation factor 4E-1 | 0.0112 | 0.4691 | 1 |
Schistosoma mansoni | hypothetical protein | 0.0016 | 0.0428 | 0.0506 |
Echinococcus granulosus | Basic leucine zipper bZIP transcription | 0.0035 | 0.1282 | 0.1729 |
Trichomonas vaginalis | eukaryotic translation initiation factor 4E, putative | 0.0112 | 0.4691 | 0.4691 |
Echinococcus multilocularis | Ataxin 2, N terminal,domain containing protein | 0.0011 | 0.021 | 0.0193 |
Plasmodium falciparum | ataxin-2 like protein, putative | 0.0025 | 0.0814 | 1 |
Schistosoma mansoni | transcription factor LCR-F1 | 0.0035 | 0.1282 | 0.1729 |
Leishmania major | hypothetical protein, conserved | 0.0025 | 0.0814 | 0.1147 |
Entamoeba histolytica | hypothetical protein | 0.0035 | 0.1282 | 0.2216 |
Loa Loa (eye worm) | hypothetical protein | 0.003 | 0.1038 | 0.1031 |
Schistosoma mansoni | histone-lysine n-methyltransferase setb1 | 0.003 | 0.1038 | 0.138 |
Trichomonas vaginalis | eukaryotic translation initiation factor 4E, putative | 0.0112 | 0.4691 | 0.4691 |
Echinococcus granulosus | cadherin EGF LAG seven pass G type receptor | 0.0016 | 0.0428 | 0.0506 |
Schistosoma mansoni | histone-lysine n-methyltransferase setb1 | 0.003 | 0.1038 | 0.138 |
Schistosoma mansoni | hypothetical protein | 0.0016 | 0.0428 | 0.0506 |
Trichomonas vaginalis | eukaryotic translation initiation factor 4E, putative | 0.0112 | 0.4691 | 0.4691 |
Leishmania major | eukaryotic translation initiation factor-like protein | 0.0112 | 0.4691 | 1 |
Plasmodium falciparum | AP endonuclease (DNA-[apurinic or apyrimidinic site] lyase), putative | 0.0018 | 0.0532 | 0.4405 |
Entamoeba histolytica | eukaryotic translation initiation factor 4E, putative | 0.0112 | 0.4691 | 1 |
Schistosoma mansoni | Guanine nucleotide-binding protein G(s) subunit alpha (Adenylate cyclase-stimulating G alpha protein) | 0.0045 | 0.1706 | 0.2337 |
Brugia malayi | hypothetical protein | 0.0016 | 0.0425 | 0.0325 |
Loa Loa (eye worm) | translation initiation factor 4E | 0.0112 | 0.4691 | 0.5277 |
Echinococcus multilocularis | eukaryotic translation initiation factor 4E | 0.0112 | 0.4691 | 0.6614 |
Echinococcus granulosus | eukaryotic translation initiation factor 4E type | 0.0013 | 0.0311 | 0.0339 |
Onchocerca volvulus | 0.0028 | 0.0962 | 0.0671 | |
Schistosoma mansoni | hypothetical protein | 0.0035 | 0.1252 | 0.1687 |
Trichomonas vaginalis | eukaryotic translation initiation factor 4E type, putative | 0.0013 | 0.0311 | 0.0311 |
Brugia malayi | exodeoxyribonuclease III family protein | 0.0018 | 0.0532 | 0.0449 |
Trichomonas vaginalis | ap endonuclease, putative | 0.0018 | 0.0532 | 0.0532 |
Schistosoma mansoni | hypothetical protein | 0.0016 | 0.0428 | 0.0506 |
Echinococcus granulosus | 5'partial|histone lysine N methyltransferase SETDB2 | 0.0028 | 0.0963 | 0.1273 |
Toxoplasma gondii | exonuclease III APE | 0.0018 | 0.0532 | 0.0505 |
Brugia malayi | translation initiation factor 4E | 0.0112 | 0.4691 | 0.5279 |
Trichomonas vaginalis | eukaryotic translation initiation factor 4E, putative | 0.0013 | 0.0311 | 0.0311 |
Trichomonas vaginalis | eukaryotic translation initiation factor 4E, putative | 0.0013 | 0.0311 | 0.0311 |
Plasmodium vivax | AP endonuclease (DNA-[apurinic or apyrimidinic site] lyase), putative | 0.0018 | 0.0532 | 0.3046 |
Trichomonas vaginalis | eukaryotic translation initiation factor 4E, putative | 0.0013 | 0.0311 | 0.0311 |
Echinococcus granulosus | DNA apurinic or apyrimidinic site lyase | 0.0018 | 0.0532 | 0.0656 |
Toxoplasma gondii | LsmAD domain-containing protein | 0.0025 | 0.0814 | 0.1147 |
Echinococcus multilocularis | diuretic hormone 44 receptor GPRdih2 | 0.0016 | 0.0428 | 0.0506 |
Echinococcus granulosus | geminin | 0.0166 | 0.7054 | 1 |
Schistosoma mansoni | histone-lysine n-methyltransferase setb1 | 0.003 | 0.1038 | 0.138 |
Echinococcus granulosus | guanine nucleotide binding protein Gs subunit | 0.0045 | 0.1706 | 0.2337 |
Brugia malayi | calcium-independent alpha-latrotoxin receptor 2, putative | 0.0016 | 0.0428 | 0.0328 |
Trichomonas vaginalis | eukaryotic translation initiation factor 4E, putative | 0.0013 | 0.0311 | 0.0311 |
Trypanosoma brucei | Eukaryotic translation initiation factor 4E-1 | 0.0112 | 0.4691 | 1 |
Plasmodium falciparum | ataxin-2 like protein, putative | 0.0025 | 0.0814 | 1 |
Leishmania major | apurinic/apyrimidinic endonuclease-redox protein | 0.0018 | 0.0532 | 0.0505 |
Brugia malayi | Corticotropin releasing factor receptor 2 precursor, putative | 0.0051 | 0.1962 | 0.2109 |
Brugia malayi | CXXC zinc finger family protein | 0.0028 | 0.0962 | 0.0948 |
Schistosoma mansoni | cpg binding protein | 0.003 | 0.1032 | 0.1372 |
Trichomonas vaginalis | ap endonuclease, putative | 0.0018 | 0.0532 | 0.0532 |
Brugia malayi | hypothetical protein | 0.0035 | 0.1282 | 0.1319 |
Trichomonas vaginalis | eukaryotic translation initiation factor 4E, putative | 0.0013 | 0.0311 | 0.0311 |
Entamoeba histolytica | hypothetical protein | 0.0035 | 0.1282 | 0.2216 |
Echinococcus granulosus | eukaryotic translation initiation factor 4E | 0.0112 | 0.4691 | 0.6614 |
Loa Loa (eye worm) | CXXC zinc finger family protein | 0.0028 | 0.0962 | 0.0943 |
Trypanosoma brucei | apurinic/apyrimidinic endonuclease, putative | 0.0018 | 0.0532 | 0.0505 |
Schistosoma mansoni | eukaryotic translation initiation factor 4e | 0.0112 | 0.4691 | 0.6614 |
Plasmodium vivax | SET domain protein, putative | 0.003 | 0.1038 | 1 |
Trypanosoma cruzi | PAB1-binding protein , putative | 0.0025 | 0.0814 | 0.1147 |
Echinococcus granulosus | histone lysine methyltransferase setb | 0.003 | 0.1038 | 0.138 |
Schistosoma mansoni | Guanine nucleotide-binding protein G(s) subunit alpha (Adenylate cyclase-stimulating G alpha protein) | 0.0045 | 0.1706 | 0.2337 |
Trypanosoma cruzi | PAB1-binding protein , putative | 0.0025 | 0.0814 | 0.1147 |
Echinococcus multilocularis | guanine nucleotide binding protein G(s) subunit | 0.0045 | 0.1706 | 0.2337 |
Brugia malayi | Calcitonin receptor-like protein seb-1 | 0.0051 | 0.1962 | 0.2109 |
Plasmodium vivax | ataxin-2 like protein, putative | 0.0025 | 0.0814 | 0.6914 |
Mycobacterium ulcerans | exodeoxyribonuclease III protein XthA | 0.0018 | 0.0532 | 0.5 |
Trichomonas vaginalis | conserved hypothetical protein | 0.0013 | 0.0311 | 0.0311 |
Echinococcus multilocularis | cadherin EGF LAG seven pass G type receptor | 0.0016 | 0.0428 | 0.0506 |
Echinococcus multilocularis | DNA (apurinic or apyrimidinic site) lyase | 0.0018 | 0.0532 | 0.0656 |
Entamoeba histolytica | hypothetical protein | 0.0035 | 0.1282 | 0.2216 |
Entamoeba histolytica | eukaryotic translation initiation factor 4E, putative | 0.0112 | 0.4691 | 1 |
Echinococcus granulosus | histone lysine N methyltransferase MLL3 | 0.001 | 0.0151 | 0.0109 |
Echinococcus multilocularis | Basic leucine zipper (bZIP) transcription | 0.0035 | 0.1282 | 0.1729 |
Schistosoma mansoni | cpg binding protein | 0.0028 | 0.0962 | 0.1271 |
Brugia malayi | Pre-SET motif family protein | 0.003 | 0.1038 | 0.1036 |
Schistosoma mansoni | hypothetical protein | 0.0166 | 0.7054 | 1 |
Echinococcus granulosus | Ataxin 2 N terminaldomain containing protein | 0.0011 | 0.021 | 0.0193 |
Trichomonas vaginalis | eukaryotic translation initiation factor 4E, putative | 0.0013 | 0.0311 | 0.0311 |
Loa Loa (eye worm) | pre-SET domain-containing protein family protein | 0.0204 | 0.8755 | 1 |
Echinococcus granulosus | guanine nucleotide binding protein Gs subunit | 0.0045 | 0.1706 | 0.2337 |
Trichomonas vaginalis | eukaryotic translation initiation factor 4E type, putative | 0.0013 | 0.0311 | 0.0311 |
Brugia malayi | hypothetical protein | 0.0025 | 0.0814 | 0.0776 |
Loa Loa (eye worm) | pigment dispersing factor receptor c | 0.0051 | 0.1962 | 0.2105 |
Schistosoma mansoni | Guanine nucleotide-binding protein G(s) subunit alpha (Adenylate cyclase-stimulating G alpha protein) | 0.0045 | 0.1706 | 0.2337 |
Giardia lamblia | Endonuclease/Exonuclease/phosphatase | 0.0018 | 0.0532 | 1 |
Trichomonas vaginalis | conserved hypothetical protein | 0.0013 | 0.0311 | 0.0311 |
Schistosoma mansoni | ap endonuclease | 0.0018 | 0.0532 | 0.0656 |
Echinococcus multilocularis | guanine nucleotide binding protein G(s) subunit | 0.0045 | 0.1706 | 0.2337 |
Trichomonas vaginalis | hypothetical protein | 0.0013 | 0.0311 | 0.0311 |
Trypanosoma cruzi | apurinic/apyrimidinic endonuclease, putative | 0.0018 | 0.0532 | 0.0505 |
Trichomonas vaginalis | eukaryotic translation initiation factor 4E type, putative | 0.0013 | 0.0311 | 0.0311 |
Toxoplasma gondii | histone lysine methyltransferase SET1 | 0.0054 | 0.2121 | 0.4133 |
Trypanosoma cruzi | Eukaryotic translation initiation factor 4E-1 | 0.0112 | 0.4691 | 1 |
Echinococcus multilocularis | cpg binding protein | 0.003 | 0.1032 | 0.1372 |
Toxoplasma gondii | histone lysine methyltransferase SET/SUV39 | 0.003 | 0.1038 | 0.1659 |
Trypanosoma brucei | PAB1-binding protein , putative | 0.0025 | 0.0814 | 0.1147 |
Loa Loa (eye worm) | exodeoxyribonuclease III family protein | 0.0018 | 0.0532 | 0.0444 |
Loa Loa (eye worm) | hypothetical protein | 0.0051 | 0.1962 | 0.2105 |
Brugia malayi | Pre-SET motif family protein | 0.0204 | 0.8755 | 1 |
Entamoeba histolytica | hypothetical protein | 0.0035 | 0.1282 | 0.2216 |
Toxoplasma gondii | eukaryotic initiation factor-4E, putative | 0.0112 | 0.4691 | 1 |
Trichomonas vaginalis | eukaryotic translation initiation factor 4E, putative | 0.0112 | 0.4691 | 0.4691 |
Trypanosoma cruzi | apurinic/apyrimidinic endonuclease | 0.0018 | 0.0532 | 0.0505 |
Loa Loa (eye worm) | hypothetical protein | 0.0016 | 0.0428 | 0.0323 |
Schistosoma mansoni | hypothetical protein | 0.0035 | 0.1282 | 0.1729 |
Schistosoma mansoni | hypothetical protein | 0.0016 | 0.0428 | 0.0506 |
Echinococcus multilocularis | histone lysine N methyltransferase MLL3 | 0.001 | 0.0151 | 0.0109 |
Loa Loa (eye worm) | GTP-binding regulatory protein Gs alpha-S chain | 0.0045 | 0.1706 | 0.1807 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
P | = 0.01 M l-1 | Partition coefficient(P) of the compound in octanol/water system | ChEMBL. | 10571171 |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.
1 literature reference was collected for this gene.