Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Plasmodium falciparum | glutamine--fructose-6-phosphate aminotransferase [isomerizing], putative | 0.002 | 0.0124 | 0.0049 |
Mycobacterium ulcerans | 6-phosphogluconate dehydrogenase | 0.0696 | 1 | 1 |
Loa Loa (eye worm) | hypothetical protein | 0.0068 | 0.082 | 0.0705 |
Leishmania major | 6-phosphogluconate dehydrogenase, decarboxylating, putative | 0.0696 | 1 | 1 |
Trypanosoma cruzi | carnitine/choline acetyltransferase, putative | 0.0029 | 0.0264 | 0.0142 |
Trypanosoma cruzi | choline/carnitine O-acyltransferase, putative | 0.0131 | 0.1742 | 0.1638 |
Schistosoma mansoni | choline o-acyltransferase | 0.0068 | 0.082 | 0.0705 |
Trypanosoma cruzi | 6-phosphogluconate dehydrogenase, decarboxylating | 0.0415 | 0.589 | 0.5838 |
Trypanosoma brucei | carnitine O-palmitoyltransferase II, putative | 0.0029 | 0.0264 | 0.0142 |
Trypanosoma cruzi | hypothetical protein, conserved | 0.0029 | 0.0264 | 0.0142 |
Trypanosoma cruzi | N-myristoyl transferase, putative | 0.004 | 0.0419 | 0.0299 |
Mycobacterium leprae | PROBABLE NAPHTHOATE SYNTHASE MENB (DIHYDROXYNAPHTHOIC ACID SYNTHETASE) (DHNA SYNTHETASE) | 0.0199 | 0.2744 | 0.2653 |
Trichomonas vaginalis | 3-hydroxyisobutyrate dehydrogenase, putative | 0.0696 | 1 | 1 |
Toxoplasma gondii | glucosamine-fructose-6-phosphate aminotransferase | 0.002 | 0.0124 | 0.0017 |
Entamoeba histolytica | glycylpeptide N-tetradecanoyltransferase, putative | 0.004 | 0.0419 | 1 |
Echinococcus granulosus | CREB binding protein | 0.007 | 0.086 | 0.086 |
Trypanosoma cruzi | choline/carnitine O-acetyltransferase, putative | 0.0029 | 0.0264 | 0.0142 |
Trypanosoma brucei | Mitochondrial SSU ribosomal protein, putative | 0.0085 | 0.1081 | 0.0969 |
Giardia lamblia | 6-phosphogluconate dehydrogenase, decarboxylating | 0.0696 | 1 | 1 |
Trypanosoma brucei | carnitine O-acetyltransferase, putative | 0.0029 | 0.0264 | 0.0142 |
Echinococcus granulosus | glycylpeptide N tetradecanoyltransferase | 0.004 | 0.0419 | 0.0419 |
Trypanosoma cruzi | carnitine/choline acetyltransferase, putative | 0.0029 | 0.0264 | 0.0142 |
Mycobacterium ulcerans | 6-phosphogluconate dehydrogenase | 0.0696 | 1 | 1 |
Echinococcus granulosus | carnitine O palmitoyltransferase 2 | 0.0029 | 0.0264 | 0.0264 |
Loa Loa (eye worm) | CBP-B | 0.0049 | 0.0551 | 0.0433 |
Trypanosoma brucei | N-myristoyl transferase, putative | 0.004 | 0.0419 | 0.0299 |
Onchocerca volvulus | 0.0029 | 0.0264 | 1 | |
Schistosoma mansoni | choline o-acyltransferase | 0.0029 | 0.0264 | 0.0142 |
Trichomonas vaginalis | glucosamine-fructose-6-phosphate aminotransferase, putative | 0.002 | 0.0124 | 0.0017 |
Entamoeba histolytica | glucosamine--fructose-6-phosphate aminotransferase, putative | 0.002 | 0.0124 | 0.1425 |
Brugia malayi | acetyltransferase, GNAT family protein | 0.0047 | 0.0523 | 0.0404 |
Schistosoma mansoni | CREB-binding protein 2 | 0.007 | 0.086 | 0.0745 |
Leishmania major | 2-hydroxy-3-oxopropionate reductase, putative | 0.0085 | 0.1081 | 0.0969 |
Trichomonas vaginalis | amidophosphoribosyltransferase, putative | 0.002 | 0.0124 | 0.0017 |
Plasmodium falciparum | 6-phosphogluconate dehydrogenase, decarboxylating, putative | 0.0696 | 1 | 1 |
Trichomonas vaginalis | glucosamine-fructose-6-phosphate aminotransferase, putative | 0.002 | 0.0124 | 0.0017 |
Loa Loa (eye worm) | acetyltransferase | 0.0047 | 0.0523 | 0.0404 |
Echinococcus multilocularis | choline O acetyltransferase | 0.0068 | 0.082 | 0.082 |
Loa Loa (eye worm) | choline/Carnitine O-acyltransferase | 0.0029 | 0.0264 | 0.0142 |
Echinococcus multilocularis | gcn5proteinral control of amino acid synthesis | 0.0047 | 0.0523 | 0.0523 |
Trypanosoma brucei | N-myristoyltransferase | 0.004 | 0.0419 | 0.0299 |
Trypanosoma cruzi | hypothetical protein, conserved | 0.0029 | 0.0264 | 0.0142 |
Trypanosoma cruzi | N-myristoyl transferase, putative | 0.004 | 0.0419 | 0.0299 |
Mycobacterium tuberculosis | Probable 6-phosphogluconate dehydrogenase Gnd1 | 0.0696 | 1 | 1 |
Loa Loa (eye worm) | choline O-acetyltransferase | 0.0068 | 0.082 | 0.0705 |
Trypanosoma cruzi | hypothetical protein, conserved | 0.0029 | 0.0264 | 0.0142 |
Trypanosoma cruzi | hypothetical protein, conserved | 0.0029 | 0.0264 | 0.0142 |
Schistosoma mansoni | CREB-binding protein 1 (SmCBP1) | 0.007 | 0.086 | 0.0745 |
Onchocerca volvulus | 0.0029 | 0.0264 | 1 | |
Leishmania major | N-myristoyl transferase, putative | 0.004 | 0.0419 | 0.0299 |
Mycobacterium tuberculosis | Naphthoate synthase MenB (dihydroxynaphthoic acid synthetase) (DHNA synthetase) | 0.0199 | 0.2744 | 0.1864 |
Echinococcus multilocularis | carnitine O palmitoyltransferase 1, liver | 0.0131 | 0.1742 | 0.1742 |
Toxoplasma gondii | 3-hydroxyisobutyrate dehydrogenase | 0.0085 | 0.1081 | 0.0985 |
Plasmodium falciparum | glycylpeptide N-tetradecanoyltransferase | 0.004 | 0.0419 | 0.0347 |
Trypanosoma brucei | 2-hydroxy-3-oxopropionate reductase, putative | 0.0085 | 0.1081 | 0.0969 |
Echinococcus multilocularis | carnitine O palmitoyltransferase 2 | 0.0029 | 0.0264 | 0.0264 |
Trypanosoma cruzi | 2-hydroxy-3-oxopropionate reductase, putative | 0.0085 | 0.1081 | 0.0969 |
Brugia malayi | Choline O-acetyltransferase | 0.0068 | 0.082 | 0.0705 |
Loa Loa (eye worm) | hypothetical protein | 0.0033 | 0.0309 | 0.0187 |
Toxoplasma gondii | 6-phosphogluconate dehydrogenase | 0.0696 | 1 | 1 |
Schistosoma mansoni | 6-phosphogluconate dehydrogenase | 0.0696 | 1 | 1 |
Echinococcus granulosus | histone acetyltransferase KAT2B | 0.0019 | 0.0107 | 0.0107 |
Schistosoma mansoni | N-myristoyltransferase | 0.004 | 0.0419 | 0.0299 |
Trypanosoma cruzi | NAD binding domain of 6-phosphogluconate dehydrogenase/NAD-binding of NADP-dependent 3-hydroxyisobutyrate dehydrogenase, putativ | 0.0085 | 0.1081 | 0.0969 |
Plasmodium vivax | glycylpeptide N-tetradecanoyltransferase, putative | 0.004 | 0.0419 | 0.0316 |
Trypanosoma cruzi | 6-phosphogluconate dehydrogenase, decarboxylating, putative | 0.0696 | 1 | 1 |
Mycobacterium tuberculosis | Probable 6-phosphogluconate dehydrogenase, decarboxylating Gnd2 | 0.0696 | 1 | 1 |
Giardia lamblia | CDC72 | 0.004 | 0.0419 | 0.0347 |
Schistosoma mansoni | transcription initiation factor iia (tfiia) gamma chain | 0.0282 | 0.3944 | 0.3868 |
Chlamydia trachomatis | GutQ/KpsF family sugar-phosphate isomerase | 0.0277 | 0.3878 | 0.3801 |
Leishmania major | dehydrogenase-like protein | 0.0085 | 0.1081 | 0.0969 |
Plasmodium vivax | glutamine--fructose-6-phosphate aminotransferase [isomerizing], putative | 0.002 | 0.0124 | 0.0017 |
Echinococcus multilocularis | glycylpeptide N tetradecanoyltransferase | 0.004 | 0.0419 | 0.0419 |
Brugia malayi | Choline/Carnitine o-acyltransferase family protein | 0.0029 | 0.0264 | 0.0142 |
Trypanosoma cruzi | choline/carnitine O-acyltransferase, putative | 0.0131 | 0.1742 | 0.1638 |
Brugia malayi | Choline O-acetyltransferase | 0.0068 | 0.082 | 0.0705 |
Trichomonas vaginalis | N-myristoyl transferase, putative | 0.004 | 0.0419 | 0.0316 |
Trypanosoma cruzi | NAD binding domain of 6-phosphogluconate dehydrogenase/NAD-binding of NADP-dependent 3-hydroxyisobutyrate dehydrogenase, putativ | 0.0085 | 0.1081 | 0.0969 |
Plasmodium vivax | 6-phosphogluconate dehydrogenase, decarboxylating, putative | 0.0696 | 1 | 1 |
Echinococcus granulosus | carnitine O palmitoyltransferase 1 liver | 0.0131 | 0.1742 | 0.1742 |
Echinococcus granulosus | Glutamine:fructose 6 phosphate aminotransferase | 0.002 | 0.0124 | 0.0124 |
Onchocerca volvulus | 0.0029 | 0.0264 | 1 | |
Brugia malayi | Choline/Carnitine o-acyltransferase family protein | 0.0204 | 0.2817 | 0.2727 |
Mycobacterium leprae | PROBABLE 6-PHOSPHOGLUCONATE DEHYDROGENASE GND1 | 0.0696 | 1 | 1 |
Leishmania major | carnitine/choline acetyltransferase, putative | 0.0029 | 0.0264 | 0.0142 |
Trichomonas vaginalis | 6-phosphogluconate dehydrogenase, putative | 0.0696 | 1 | 1 |
Loa Loa (eye worm) | pgd protein | 0.0696 | 1 | 1 |
Trypanosoma brucei | carnitine O-palmitoyltransferase, putative | 0.0029 | 0.0264 | 0.0142 |
Echinococcus multilocularis | Glutamine:fructose 6 phosphate aminotransferase | 0.002 | 0.0124 | 0.0124 |
Schistosoma mansoni | gcn5proteinral control of amino-acid synthesis 5-like 2 gcnl2 | 0.0047 | 0.0523 | 0.0404 |
Trypanosoma cruzi | carnitine O-palmitoyltransferase II, putative | 0.0029 | 0.0264 | 0.0142 |
Mycobacterium ulcerans | 3-hydroxyisobutyrate dehydrogenase | 0.0085 | 0.1081 | 0.0969 |
Leishmania major | choline/Carnitine o-acyltransferase-like protein | 0.0131 | 0.1742 | 0.1638 |
Toxoplasma gondii | 6-phosphogluconate dehydrogenase | 0.0696 | 1 | 1 |
Trypanosoma brucei | hypothetical protein, conserved | 0.0029 | 0.0264 | 0.0142 |
Echinococcus granulosus | histone acetyltransferase KAT2B | 0.0039 | 0.0407 | 0.0407 |
Echinococcus granulosus | CREB binding protein | 0.0044 | 0.0472 | 0.0472 |
Loa Loa (eye worm) | carnitine O-palmitoyltransferase I isoform | 0.0029 | 0.0264 | 0.0142 |
Loa Loa (eye worm) | N-myristoyltransferase 2 | 0.004 | 0.0419 | 0.0299 |
Trypanosoma brucei | 6-phosphogluconate dehydrogenase, decarboxylating | 0.0696 | 1 | 1 |
Loa Loa (eye worm) | hypothetical protein | 0.0204 | 0.2817 | 0.2727 |
Echinococcus multilocularis | CREB binding protein | 0.0049 | 0.0542 | 0.0542 |
Echinococcus granulosus | 6 phosphogluconate dehydrogenase | 0.0696 | 1 | 1 |
Trypanosoma cruzi | choline/carnitine O-acyltransferase, putative | 0.0029 | 0.0264 | 0.0142 |
Trypanosoma cruzi | 6-phosphogluconate dehydrogenase, decarboxylating, putative | 0.0282 | 0.3944 | 0.3868 |
Brugia malayi | TAZ zinc finger family protein | 0.007 | 0.086 | 0.0745 |
Mycobacterium ulcerans | naphthoate synthase | 0.0199 | 0.2744 | 0.2653 |
Trichomonas vaginalis | 6-phosphogluconate dehydrogenase, putative | 0.0696 | 1 | 1 |
Chlamydia trachomatis | 6-phosphogluconate dehydrogenase | 0.0696 | 1 | 1 |
Treponema pallidum | 6-phosphogluconate dehydrogenase | 0.0696 | 1 | 1 |
Trichomonas vaginalis | N-myristoyl transferase, putative | 0.0026 | 0.0219 | 0.0113 |
Echinococcus granulosus | choline O acetyltransferase | 0.0068 | 0.082 | 0.082 |
Leishmania major | carnitine palmitoyltransferase-like protein | 0.0029 | 0.0264 | 0.0142 |
Trypanosoma cruzi | hypothetical protein, conserved | 0.0029 | 0.0264 | 0.0142 |
Brugia malayi | N-myristoyltransferase 2 | 0.004 | 0.0419 | 0.0299 |
Echinococcus multilocularis | 6 phosphogluconate dehydrogenase | 0.0696 | 1 | 1 |
Onchocerca volvulus | 0.0029 | 0.0264 | 1 | |
Toxoplasma gondii | phosphogluconate dehydrogenase (decarboxylating), NAD binding domain-containing protein | 0.0085 | 0.1081 | 0.0985 |
Wolbachia endosymbiont of Brugia malayi | glucosamine 6-phosphate synthetase | 0.002 | 0.0124 | 0.5 |
Brugia malayi | Choline/Carnitine o-acyltransferase family protein | 0.0029 | 0.0264 | 0.0142 |
Trypanosoma cruzi | 2-hydroxy-3-oxopropionate reductase, putative | 0.0085 | 0.1081 | 0.0969 |
Trypanosoma cruzi | carnitine O-acetyltransferase, putative | 0.0029 | 0.0264 | 0.0142 |
Trypanosoma brucei | carnitine O-palmitoyltransferase II, putative | 0.0029 | 0.0264 | 0.0142 |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.