Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Trypanosoma cruzi | trans-sialidase, putative | 0.0033 | 0.7062 | 0.6755 |
Trichomonas vaginalis | multidrug resistance protein 1, 2, putative | 0.0014 | 0.1753 | 0.1753 |
Trichomonas vaginalis | abcb9, putative | 0.0014 | 0.1753 | 0.1753 |
Entamoeba histolytica | ABC transporter, putative | 0.0018 | 0.2763 | 0.1224 |
Loa Loa (eye worm) | ATP-binding cassette sub-family B member 2 | 0.0014 | 0.1753 | 0.0828 |
Leishmania major | ubiquitin-conjugating enzyme e2, putative | 0.0044 | 1 | 1 |
Trypanosoma cruzi | trans-sialidase, putative | 0.0033 | 0.7062 | 0.6755 |
Giardia lamblia | Multidrug resistance-associated protein 1 | 0.0018 | 0.2763 | 1 |
Loa Loa (eye worm) | ubiquitin conjugating enzyme protein 13 | 0.0044 | 1 | 1 |
Trypanosoma brucei | trans-sialidase | 0.0033 | 0.7063 | 0.5942 |
Trichomonas vaginalis | multidrug resistance protein 1, 2, putative | 0.0014 | 0.1753 | 0.1753 |
Chlamydia trachomatis | ABC transporter ATP binding protein/permease | 0.0014 | 0.1753 | 0.5 |
Leishmania major | ATP-binding cassette protein subfamily C, member 5, putative | 0.0018 | 0.2763 | 0.1224 |
Brugia malayi | multidrug resistance related protein 1 | 0.0018 | 0.2763 | 0.1224 |
Trypanosoma cruzi | trans-sialidase, putative | 0.0033 | 0.7062 | 0.6755 |
Trypanosoma cruzi | trans-sialidase, putative | 0.0033 | 0.7063 | 0.6756 |
Trichomonas vaginalis | abcb9, putative | 0.0014 | 0.1753 | 0.1753 |
Trichomonas vaginalis | lipid A export ATP-binding/permease protein msba, putative | 0.0014 | 0.1753 | 0.1753 |
Trypanosoma cruzi | trans-sialidase, putative | 0.0033 | 0.7063 | 0.6756 |
Trichomonas vaginalis | multidrug resistance protein 1, 2, putative | 0.0014 | 0.1753 | 0.1753 |
Echinococcus multilocularis | ATP binding cassette subfamily B (MDR:TAP) | 0.0014 | 0.1753 | 0.1753 |
Trypanosoma brucei | trans-sialidase, putative | 0.0033 | 0.7063 | 0.5942 |
Trypanosoma brucei | trans-sialidase, putative | 0.0033 | 0.7063 | 0.5942 |
Trichomonas vaginalis | ATP-binding cassette transporter, putative | 0.0014 | 0.1753 | 0.1753 |
Trypanosoma cruzi | trans-sialidase, Group I, putative | 0.0033 | 0.7063 | 0.6756 |
Trypanosoma cruzi | ubiquitin-conjugating enzyme E2, putative | 0.0044 | 1 | 1 |
Trichomonas vaginalis | abcb9, putative | 0.0014 | 0.1753 | 0.1753 |
Trichomonas vaginalis | ubiquitin-conjugating enzyme E2, putative | 0.0044 | 1 | 1 |
Leishmania major | p-glycoprotein e | 0.0018 | 0.2763 | 0.1224 |
Schistosoma mansoni | multidrug resistance protein | 0.0018 | 0.2763 | 0.1224 |
Entamoeba histolytica | hypothetical protein | 0.0018 | 0.2763 | 0.1224 |
Echinococcus granulosus | ubiquitin conjugating enzyme E2 N | 0.0044 | 1 | 1 |
Loa Loa (eye worm) | hypothetical protein | 0.0018 | 0.2763 | 0.195 |
Trichomonas vaginalis | lipid A export ATP-binding/permease protein msba, putative | 0.0014 | 0.1753 | 0.1753 |
Echinococcus granulosus | ATP binding cassette subfamily B MDR:TAP | 0.0014 | 0.1753 | 0.1753 |
Trichomonas vaginalis | ABC transporter, half transporter, putative | 0.0014 | 0.1753 | 0.1753 |
Leishmania major | ABC-thiol transporter | 0.0018 | 0.2763 | 0.1224 |
Echinococcus multilocularis | multidrug resistance protein 1 | 0.0014 | 0.1753 | 0.1753 |
Trypanosoma brucei | trans-sialidase, putative | 0.0033 | 0.7063 | 0.5942 |
Trypanosoma cruzi | trans-sialidase, Group I, putative | 0.0033 | 0.7063 | 0.6756 |
Loa Loa (eye worm) | multidrug resistance protein 3 | 0.0014 | 0.1753 | 0.0828 |
Trypanosoma cruzi | trans-sialidase, Group I, putative | 0.0033 | 0.7063 | 0.6756 |
Brugia malayi | ABC transporter transmembrane region family protein | 0.0018 | 0.2763 | 0.1224 |
Loa Loa (eye worm) | hypothetical protein | 0.0017 | 0.2699 | 0.188 |
Leishmania major | ATP-binding cassette protein subfamily C, member 2, putative | 0.0018 | 0.2763 | 0.1224 |
Trypanosoma brucei | ubiquitin-protein ligase, putative | 0.0044 | 1 | 1 |
Loa Loa (eye worm) | hypothetical protein | 0.0014 | 0.169 | 0.0757 |
Leishmania major | ATP-binding cassette protein subfamily C, member 1, putative | 0.0018 | 0.2763 | 0.1224 |
Schistosoma mansoni | ubiquitin conjugating enzyme 13 | 0.0044 | 1 | 1 |
Loa Loa (eye worm) | hypothetical protein | 0.0018 | 0.2763 | 0.195 |
Echinococcus granulosus | multidrug resistance protein 1 | 0.0014 | 0.1753 | 0.1753 |
Entamoeba histolytica | ATP-binding cassette protein, putative | 0.0018 | 0.2763 | 0.1224 |
Echinococcus multilocularis | ATP binding cassette subfamily B (MDR:TAP) | 0.0014 | 0.1753 | 0.1753 |
Trypanosoma cruzi | multidrug resistance-associated protein, putative | 0.0018 | 0.2763 | 0.2006 |
Schistosoma mansoni | multidrug resistance protein | 0.0018 | 0.2763 | 0.1224 |
Trypanosoma brucei | trans-sialidase, putative | 0.0033 | 0.7063 | 0.5942 |
Trichomonas vaginalis | lipid A export ATP-binding/permease protein msba, putative | 0.0014 | 0.1753 | 0.1753 |
Mycobacterium tuberculosis | Probable transmembrane multidrug efflux pump | 0.0014 | 0.1753 | 0.5 |
Trypanosoma cruzi | trans-sialidase, Group I, putative | 0.0033 | 0.7063 | 0.6756 |
Trichomonas vaginalis | multidrug resistance protein 1, 2, putative | 0.0014 | 0.1753 | 0.1753 |
Trypanosoma brucei | trans-sialidase, putative | 0.0033 | 0.7063 | 0.5942 |
Echinococcus multilocularis | multidrug resistance associated protein 7 | 0.0018 | 0.2763 | 0.2763 |
Loa Loa (eye worm) | ubiquitin conjugating enzyme protein 13 | 0.0044 | 1 | 1 |
Echinococcus multilocularis | ATP binding cassette sub family B | 0.0014 | 0.169 | 0.169 |
Echinococcus granulosus | multidrug resistance associated protein 1 | 0.0018 | 0.2763 | 0.2763 |
Echinococcus granulosus | ATP binding cassette subfamily B MDR:TAP | 0.0014 | 0.1753 | 0.1753 |
Trichomonas vaginalis | multidrug resistance protein 1, 2, putative | 0.0014 | 0.1753 | 0.1753 |
Trichomonas vaginalis | lipid A export ATP-binding/permease protein msba, putative | 0.0014 | 0.1753 | 0.1753 |
Trichomonas vaginalis | ATP-binding cassette transporter, putative | 0.0014 | 0.1753 | 0.1753 |
Toxoplasma gondii | ubiquitin-conjugating enzyme subfamily protein | 0.0044 | 1 | 1 |
Trichomonas vaginalis | lipid A export ATP-binding/permease protein msba, putative | 0.0014 | 0.1753 | 0.1753 |
Schistosoma mansoni | multidrug resistance protein | 0.0018 | 0.2763 | 0.1224 |
Echinococcus granulosus | multidrug resistance protein 1 | 0.0014 | 0.1753 | 0.1753 |
Echinococcus multilocularis | ATP binding cassette subfamily B (MDR:TAP) | 0.0014 | 0.1753 | 0.1753 |
Loa Loa (eye worm) | hypothetical protein | 0.0014 | 0.1753 | 0.0828 |
Echinococcus granulosus | multidrug resistance associated protein 4 | 0.0011 | 0.0946 | 0.0946 |
Giardia lamblia | ABC transporter, putative | 0.0018 | 0.2763 | 1 |
Schistosoma mansoni | multidrug resistance protein | 0.0018 | 0.2763 | 0.1224 |
Trichomonas vaginalis | ABC transporter, putative | 0.0014 | 0.1753 | 0.1753 |
Trypanosoma cruzi | trans-sialidase, Group I, putative | 0.0033 | 0.7063 | 0.6756 |
Trypanosoma cruzi | trans-sialidase, Group I, putative | 0.0033 | 0.7063 | 0.6756 |
Echinococcus granulosus | 5'partial|ATP binding cassette sub family B | 0.0014 | 0.169 | 0.169 |
Trypanosoma cruzi | trans-sialidase, Group I, putative | 0.0033 | 0.7063 | 0.6756 |
Entamoeba histolytica | ubiquitin-conjugating enzyme family protein | 0.0044 | 1 | 1 |
Loa Loa (eye worm) | hypothetical protein | 0.0014 | 0.1753 | 0.0828 |
Trypanosoma cruzi | trans-sialidase, Group I, putative | 0.0033 | 0.7063 | 0.6756 |
Brugia malayi | ubiquitin conjugating enzyme protein 13 | 0.0044 | 1 | 1 |
Trichomonas vaginalis | ATP-binding cassette transporter, putative | 0.0014 | 0.1753 | 0.1753 |
Trypanosoma cruzi | multidrug resistance protein E, putative | 0.0018 | 0.2763 | 0.2006 |
Echinococcus granulosus | multidrug resistance protein 1 | 0.0014 | 0.1753 | 0.1753 |
Echinococcus multilocularis | ubiquitin conjugating enzyme E2 N | 0.0044 | 1 | 1 |
Trypanosoma cruzi | multidrug resistance-associated protein, putative | 0.0018 | 0.2763 | 0.2006 |
Leishmania major | pentamidine resistance protein 1 | 0.0018 | 0.2763 | 0.1224 |
Entamoeba histolytica | ATP-binding cassette protein, putative | 0.0018 | 0.2763 | 0.1224 |
Trichomonas vaginalis | lipid A export ATP-binding/permease protein msba, putative | 0.0014 | 0.1753 | 0.1753 |
Entamoeba histolytica | ATP-binding cassette protein, putative | 0.0018 | 0.2763 | 0.1224 |
Onchocerca volvulus | 0.0014 | 0.1753 | 0.5 | |
Plasmodium vivax | ubiquitin-conjugating enzyme E2 N, putative | 0.0044 | 1 | 1 |
Trichomonas vaginalis | lipid A export ATP-binding/permease protein msba, putative | 0.0014 | 0.1753 | 0.1753 |
Entamoeba histolytica | ATP-binding cassette protein, putative | 0.0018 | 0.2763 | 0.1224 |
Trypanosoma cruzi | trans-sialidase, Group I, putative | 0.0033 | 0.7063 | 0.6756 |
Trypanosoma cruzi | trans-sialidase, putative | 0.0033 | 0.7062 | 0.6755 |
Trichomonas vaginalis | taga, putative | 0.0014 | 0.1753 | 0.1753 |
Trypanosoma cruzi | trans-sialidase, putative | 0.0033 | 0.7063 | 0.6756 |
Giardia lamblia | MRP-like ABC transporter | 0.0018 | 0.2763 | 1 |
Echinococcus multilocularis | ATP binding cassette subfamily B (MDR:TAP) | 0.0014 | 0.1753 | 0.1753 |
Trichomonas vaginalis | lipid A export ATP-binding/permease protein msba, putative | 0.0014 | 0.1753 | 0.1753 |
Trypanosoma cruzi | trans-sialidase, Group I, putative | 0.0033 | 0.7063 | 0.6756 |
Echinococcus granulosus | ATP binding cassette subfamily B MDR:TAP | 0.0014 | 0.1753 | 0.1753 |
Giardia lamblia | Multidrug resistance-associated protein 1 | 0.0018 | 0.2763 | 1 |
Trichomonas vaginalis | ABC transporter, putative | 0.0014 | 0.1753 | 0.1753 |
Trichomonas vaginalis | multidrug resistance protein 1, 2, putative | 0.0014 | 0.1753 | 0.1753 |
Echinococcus multilocularis | multidrug resistance associated protein 1 | 0.0018 | 0.2763 | 0.2763 |
Leishmania major | ATP-binding cassette protein subfamily C, member 6, putative | 0.0018 | 0.2763 | 0.1224 |
Trichomonas vaginalis | ABC transporter, putative | 0.0014 | 0.1753 | 0.1753 |
Trichomonas vaginalis | multidrug resistance protein 1, 2, putative | 0.0014 | 0.1753 | 0.1753 |
Echinococcus multilocularis | multidrug resistance associated protein 4 | 0.0011 | 0.0946 | 0.0946 |
Toxoplasma gondii | ABC transporter transmembrane region domain-containing protein | 0.0018 | 0.2763 | 0.1224 |
Echinococcus granulosus | ATP binding cassette subfamily B MDR:TAP | 0.0014 | 0.1753 | 0.1753 |
Trichomonas vaginalis | ATP-binding cassette transporter, putative | 0.0014 | 0.1753 | 0.1753 |
Loa Loa (eye worm) | ABC transporter transmembrane region family protein | 0.0018 | 0.2763 | 0.195 |
Trichomonas vaginalis | ABC transporter, putative | 0.0014 | 0.1753 | 0.1753 |
Trypanosoma cruzi | ubiquitin-conjugating enzyme E2, putative | 0.0044 | 1 | 1 |
Echinococcus multilocularis | multidrug resistance protein 1 | 0.0014 | 0.1753 | 0.1753 |
Trichomonas vaginalis | ubiquitin-conjugating enzyme E2, putative | 0.0044 | 1 | 1 |
Entamoeba histolytica | multidrug resistance protein, putative | 0.0018 | 0.2763 | 0.1224 |
Trichomonas vaginalis | ATP-binding cassette transporter, putative | 0.0014 | 0.1753 | 0.1753 |
Trichomonas vaginalis | ABC transporter, half transporter, putative | 0.0014 | 0.1753 | 0.1753 |
Plasmodium falciparum | ubiquitin-conjugating enzyme E2 N, putative | 0.0044 | 1 | 1 |
Echinococcus granulosus | multidrug resistance associated protein 7 | 0.0018 | 0.2763 | 0.2763 |
Trypanosoma cruzi | trans-sialidase, Group I, putative | 0.0033 | 0.7063 | 0.6756 |
Echinococcus multilocularis | ATP binding cassette subfamily B (MDR:TAP) | 0.0014 | 0.1753 | 0.1753 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
Potency (functional) | = 25.1189 um | PUBCHEM_BIOASSAY: Secondary Concentration-Response Assay for Agonists of the Thyroid Stimulating Hormone Receptor: HTRF Activity Detection. (Class of assay: confirmatory) | ChEMBL. | No reference |
Potency (functional) | 29.0929 uM | PUBCHEM_BIOASSAY: Nrf2 qHTS screen for inhibitors. (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID493153, AID493163, AID504648] | ChEMBL. | No reference |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.