Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Trypanosoma cruzi | trans-sialidase, Group I, putative | 0.0031 | 0.6594 | 0.6594 |
Echinococcus granulosus | ubiquitin conjugating enzyme E2 N | 0.0041 | 1 | 1 |
Trypanosoma cruzi | ubiquitin-conjugating enzyme E2, putative | 0.0041 | 1 | 1 |
Trichomonas vaginalis | ATP-binding cassette transporter, putative | 0.0025 | 0.4629 | 0.3877 |
Echinococcus granulosus | multidrug resistance associated protein 7 | 0.0022 | 0.3523 | 0.3523 |
Trypanosoma cruzi | trans-sialidase, putative | 0.0031 | 0.6594 | 0.6594 |
Toxoplasma gondii | ATP-binding cassette transporter ABC.B1 | 0.0025 | 0.4629 | 0.1708 |
Entamoeba histolytica | P-glycoprotein-1 | 0.0025 | 0.4629 | 0.1708 |
Trichomonas vaginalis | ABC transporter, putative | 0.0025 | 0.4629 | 0.3877 |
Trypanosoma brucei | trans-sialidase, putative | 0.0031 | 0.6594 | 0.4741 |
Trypanosoma cruzi | trans-sialidase, Group I, putative | 0.0031 | 0.6594 | 0.6594 |
Trichomonas vaginalis | ATP-binding cassette transporter, putative | 0.0025 | 0.4629 | 0.3877 |
Brugia malayi | multidrug resistance protein 3 | 0.0025 | 0.4629 | 0.1708 |
Echinococcus multilocularis | ATP binding cassette subfamily B (MDR:TAP) | 0.0025 | 0.4629 | 0.4629 |
Echinococcus granulosus | multidrug resistance protein 1 | 0.0025 | 0.4629 | 0.4629 |
Echinococcus granulosus | multidrug resistance protein 1 | 0.0015 | 0.1229 | 0.1229 |
Echinococcus granulosus | 5'partial|ATP binding cassette sub family B | 0.0025 | 0.4506 | 0.4506 |
Trypanosoma brucei | trans-sialidase, putative | 0.0031 | 0.6594 | 0.4741 |
Trypanosoma cruzi | trans-sialidase, putative | 0.0031 | 0.6594 | 0.6594 |
Trichomonas vaginalis | taga, putative | 0.0025 | 0.4629 | 0.3877 |
Trypanosoma cruzi | trans-sialidase, Group I, putative | 0.0031 | 0.6594 | 0.6594 |
Trypanosoma cruzi | ubiquitin-conjugating enzyme E2, putative | 0.0041 | 1 | 1 |
Trypanosoma cruzi | trans-sialidase, Group I, putative | 0.0031 | 0.6594 | 0.6594 |
Trypanosoma cruzi | trans-sialidase, Group I, putative | 0.0031 | 0.6594 | 0.6594 |
Leishmania major | p-glycoprotein | 0.0025 | 0.4629 | 0.1708 |
Echinococcus granulosus | multidrug resistance protein 1 | 0.0025 | 0.4629 | 0.4629 |
Trichomonas vaginalis | ABC transporter, putative | 0.0025 | 0.4629 | 0.3877 |
Loa Loa (eye worm) | ubiquitin conjugating enzyme protein 13 | 0.0041 | 1 | 1 |
Echinococcus multilocularis | multidrug resistance protein 1 | 0.0025 | 0.4629 | 0.4629 |
Brugia malayi | ubiquitin conjugating enzyme protein 13 | 0.0041 | 1 | 1 |
Loa Loa (eye worm) | ABC transporter transmembrane region family protein | 0.0022 | 0.3523 | 0.3443 |
Echinococcus multilocularis | ATP binding cassette subfamily B (MDR:TAP) | 0.0025 | 0.4629 | 0.4629 |
Echinococcus multilocularis | multidrug resistance protein 1 | 0.0025 | 0.4629 | 0.4629 |
Loa Loa (eye worm) | hypothetical protein | 0.0025 | 0.4629 | 0.4562 |
Echinococcus multilocularis | ATP binding cassette subfamily B (MDR:TAP) | 0.0025 | 0.4629 | 0.4629 |
Trichomonas vaginalis | abcb9, putative | 0.0025 | 0.4629 | 0.3877 |
Echinococcus granulosus | ATP binding cassette subfamily B MDR:TAP | 0.0025 | 0.4629 | 0.4629 |
Trypanosoma brucei | ubiquitin-protein ligase, putative | 0.0041 | 1 | 1 |
Loa Loa (eye worm) | multidrug resistance protein 3 | 0.0025 | 0.4629 | 0.4562 |
Schistosoma mansoni | multidrug resistance protein | 0.0025 | 0.4629 | 0.1708 |
Trypanosoma brucei | trans-sialidase, putative | 0.0031 | 0.6594 | 0.4741 |
Loa Loa (eye worm) | hypothetical protein | 0.0022 | 0.3523 | 0.3443 |
Trichomonas vaginalis | lipid A export ATP-binding/permease protein msba, putative | 0.0025 | 0.4629 | 0.3877 |
Entamoeba histolytica | P-glycoprotein-5 | 0.0025 | 0.4629 | 0.1708 |
Trichomonas vaginalis | ABC transporter, putative | 0.0025 | 0.4629 | 0.3877 |
Trypanosoma brucei | trans-sialidase | 0.0031 | 0.6594 | 0.4741 |
Onchocerca volvulus | 0.0025 | 0.4629 | 0.5 | |
Trypanosoma cruzi | trans-sialidase, putative | 0.0031 | 0.6592 | 0.6592 |
Schistosoma mansoni | multidrug resistance protein | 0.0025 | 0.4629 | 0.1708 |
Mycobacterium tuberculosis | Probable transmembrane multidrug efflux pump | 0.0025 | 0.4629 | 0.5 |
Trichomonas vaginalis | lipid A export ATP-binding/permease protein msba, putative | 0.0025 | 0.4629 | 0.3877 |
Trichomonas vaginalis | lipid A export ATP-binding/permease protein msba, putative | 0.0025 | 0.4629 | 0.3877 |
Trichomonas vaginalis | ubiquitin-conjugating enzyme E2, putative | 0.0041 | 1 | 1 |
Plasmodium vivax | ubiquitin-conjugating enzyme E2 N, putative | 0.0041 | 1 | 1 |
Trichomonas vaginalis | lipid A export ATP-binding/permease protein msba, putative | 0.0025 | 0.4629 | 0.3877 |
Trypanosoma brucei | trans-sialidase, putative | 0.0031 | 0.6594 | 0.4741 |
Trypanosoma cruzi | multidrug resistance-associated protein, putative | 0.0022 | 0.3523 | 0.3523 |
Entamoeba histolytica | P-glycoprotein 5, putative | 0.0025 | 0.4629 | 0.1708 |
Leishmania major | ATP-binding cassette protein subfamily B, member 2, putative | 0.0025 | 0.4629 | 0.1708 |
Chlamydia trachomatis | ABC transporter ATP binding protein/permease | 0.0025 | 0.4629 | 0.5 |
Trichomonas vaginalis | ATP-binding cassette transporter, putative | 0.0025 | 0.4629 | 0.3877 |
Trypanosoma brucei | trans-sialidase, putative | 0.0031 | 0.6594 | 0.4741 |
Trichomonas vaginalis | multidrug resistance protein 1, 2, putative | 0.0025 | 0.4629 | 0.3877 |
Trypanosoma cruzi | trans-sialidase, Group I, putative | 0.0031 | 0.6594 | 0.6594 |
Loa Loa (eye worm) | hypothetical protein | 0.0025 | 0.4629 | 0.4562 |
Schistosoma mansoni | ubiquitin conjugating enzyme 13 | 0.0041 | 1 | 1 |
Echinococcus multilocularis | multidrug resistance protein 1 | 0.0015 | 0.1229 | 0.1229 |
Loa Loa (eye worm) | hypothetical protein | 0.0021 | 0.34 | 0.3318 |
Echinococcus granulosus | ATP binding cassette subfamily B MDR:TAP | 0.0025 | 0.4629 | 0.4629 |
Echinococcus multilocularis | multidrug resistance associated protein 7 | 0.0022 | 0.3523 | 0.3523 |
Schistosoma mansoni | multidrug resistance protein | 0.0025 | 0.4629 | 0.1708 |
Trichomonas vaginalis | lipid A export ATP-binding/permease protein msba, putative | 0.0025 | 0.4629 | 0.3877 |
Entamoeba histolytica | P-glyco protein 6, putative | 0.0025 | 0.4629 | 0.1708 |
Trichomonas vaginalis | lipid A export ATP-binding/permease protein msba, putative | 0.0025 | 0.4629 | 0.3877 |
Loa Loa (eye worm) | hypothetical protein | 0.0022 | 0.3523 | 0.3443 |
Trichomonas vaginalis | ABC transporter, half transporter, putative | 0.0025 | 0.4629 | 0.3877 |
Trypanosoma cruzi | trans-sialidase, Group I, putative | 0.0031 | 0.6594 | 0.6594 |
Trypanosoma cruzi | trans-sialidase, putative | 0.0031 | 0.6592 | 0.6592 |
Entamoeba histolytica | P-glycoprotein-2 | 0.0025 | 0.4629 | 0.1708 |
Giardia lamblia | ABC transporter, putative | 0.0022 | 0.3523 | 1 |
Trypanosoma cruzi | trans-sialidase, putative | 0.0031 | 0.6592 | 0.6592 |
Leishmania major | ubiquitin-conjugating enzyme e2, putative | 0.0041 | 1 | 1 |
Toxoplasma gondii | ABC transporter transmembrane region domain-containing protein | 0.0025 | 0.4629 | 0.1708 |
Echinococcus multilocularis | ATP binding cassette subfamily B (MDR:TAP) | 0.0025 | 0.4629 | 0.4629 |
Trypanosoma cruzi | trans-sialidase, Group I, putative | 0.0031 | 0.6594 | 0.6594 |
Entamoeba histolytica | P-glycoprotein-2 | 0.0025 | 0.4629 | 0.1708 |
Loa Loa (eye worm) | ubiquitin conjugating enzyme protein 13 | 0.0041 | 1 | 1 |
Trichomonas vaginalis | lipid A export ATP-binding/permease protein msba, putative | 0.0025 | 0.4629 | 0.3877 |
Echinococcus multilocularis | ATP binding cassette sub family B | 0.0025 | 0.4506 | 0.4506 |
Trichomonas vaginalis | multidrug resistance protein 1, 2, putative | 0.0025 | 0.4629 | 0.3877 |
Echinococcus multilocularis | multidrug resistance associated protein 1 | 0.0022 | 0.3523 | 0.3523 |
Echinococcus multilocularis | ubiquitin conjugating enzyme E2 N | 0.0041 | 1 | 1 |
Schistosoma mansoni | smdr2 | 0.0025 | 0.4629 | 0.1708 |
Trichomonas vaginalis | ABC transporter, half transporter, putative | 0.0025 | 0.4629 | 0.3877 |
Trypanosoma cruzi | trans-sialidase, putative | 0.0031 | 0.6594 | 0.6594 |
Echinococcus granulosus | ATP binding cassette subfamily B MDR:TAP | 0.0025 | 0.4629 | 0.4629 |
Trypanosoma cruzi | trans-sialidase, putative | 0.0031 | 0.6592 | 0.6592 |
Entamoeba histolytica | ubiquitin-conjugating enzyme family protein | 0.0041 | 1 | 1 |
Trichomonas vaginalis | ATP-binding cassette transporter, putative | 0.0025 | 0.4629 | 0.3877 |
Trichomonas vaginalis | multidrug resistance protein 1, 2, putative | 0.0025 | 0.4629 | 0.3877 |
Loa Loa (eye worm) | hypothetical protein | 0.0025 | 0.4506 | 0.4438 |
Trichomonas vaginalis | abcb9, putative | 0.0025 | 0.4629 | 0.3877 |
Trypanosoma cruzi | trans-sialidase, Group I, putative | 0.0031 | 0.6594 | 0.6594 |
Trypanosoma cruzi | trans-sialidase, Group I, putative | 0.0031 | 0.6594 | 0.6594 |
Trypanosoma cruzi | multidrug resistance protein E, putative | 0.0022 | 0.3523 | 0.3523 |
Trichomonas vaginalis | ATP-binding cassette transporter, putative | 0.0025 | 0.4629 | 0.3877 |
Giardia lamblia | MRP-like ABC transporter | 0.0022 | 0.3523 | 1 |
Trichomonas vaginalis | ABC transporter, putative | 0.0025 | 0.4629 | 0.3877 |
Entamoeba histolytica | P-glycoprotein-2, putative | 0.0025 | 0.4629 | 0.1708 |
Trichomonas vaginalis | abcb9, putative | 0.0025 | 0.4629 | 0.3877 |
Echinococcus granulosus | multidrug resistance protein 1 | 0.0015 | 0.1229 | 0.1229 |
Trichomonas vaginalis | lipid A export ATP-binding/permease protein msba, putative | 0.0025 | 0.4629 | 0.3877 |
Loa Loa (eye worm) | ATP-binding cassette sub-family B member 2 | 0.0025 | 0.4629 | 0.4562 |
Echinococcus granulosus | multidrug resistance associated protein 1 | 0.0022 | 0.3523 | 0.3523 |
Giardia lamblia | Multidrug resistance-associated protein 1 | 0.0022 | 0.3523 | 1 |
Trypanosoma cruzi | multidrug resistance-associated protein, putative | 0.0022 | 0.3523 | 0.3523 |
Echinococcus multilocularis | ATP binding cassette subfamily B (MDR:TAP) | 0.0025 | 0.4629 | 0.4629 |
Echinococcus granulosus | ATP binding cassette subfamily B MDR:TAP | 0.0025 | 0.4629 | 0.4629 |
Trypanosoma cruzi | trans-sialidase, Group I, putative | 0.0031 | 0.6594 | 0.6594 |
Plasmodium falciparum | ubiquitin-conjugating enzyme E2 N, putative | 0.0041 | 1 | 1 |
Trichomonas vaginalis | multidrug resistance protein 1, 2, putative | 0.0025 | 0.4629 | 0.3877 |
Trichomonas vaginalis | multidrug resistance protein 1, 2, putative | 0.0025 | 0.4629 | 0.3877 |
Trichomonas vaginalis | ubiquitin-conjugating enzyme E2, putative | 0.0041 | 1 | 1 |
Brugia malayi | ABC transporter family protein | 0.0025 | 0.4629 | 0.1708 |
Trichomonas vaginalis | multidrug resistance protein 1, 2, putative | 0.0025 | 0.4629 | 0.3877 |
Giardia lamblia | Multidrug resistance-associated protein 1 | 0.0022 | 0.3523 | 1 |
Toxoplasma gondii | ubiquitin-conjugating enzyme subfamily protein | 0.0041 | 1 | 1 |
Echinococcus granulosus | multidrug resistance protein 1 | 0.0025 | 0.4629 | 0.4629 |
Trichomonas vaginalis | multidrug resistance protein 1, 2, putative | 0.0025 | 0.4629 | 0.3877 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
IC50 (functional) | > 50 uM | Cytotoxicity against human HL60 cells after 72 hrs by MTT assay | ChEMBL. | 24095093 |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.