Species | Potential target | Raw | Global | Species |
---|---|---|---|---|
Entamoeba histolytica | P-glycoprotein-2, putative | 0.0059 | 1 | 1 |
Echinococcus granulosus | multidrug resistance protein 1 | 0.0039 | 0.4732 | 0.4732 |
Entamoeba histolytica | P-glycoprotein-2 | 0.0059 | 1 | 1 |
Toxoplasma gondii | ubiquitin-conjugating enzyme subfamily protein | 0.0042 | 0.5414 | 0.5325 |
Trypanosoma cruzi | trans-sialidase, Group I, putative | 0.0031 | 0.2812 | 0.5019 |
Trichomonas vaginalis | multidrug resistance protein 1, 2, putative | 0.0059 | 1 | 1 |
Loa Loa (eye worm) | ABC transporter | 0.0021 | 0.019 | 0.019 |
Brugia malayi | ABC transporter family protein | 0.0059 | 1 | 1 |
Trypanosoma cruzi | trans-sialidase, Group I, putative | 0.0031 | 0.2812 | 0.5019 |
Trichomonas vaginalis | abcb9, putative | 0.0059 | 1 | 1 |
Loa Loa (eye worm) | hypothetical protein | 0.0034 | 0.347 | 0.347 |
Trypanosoma cruzi | trans-sialidase, putative | 0.0031 | 0.2811 | 0.5017 |
Trypanosoma brucei | trans-sialidase | 0.0031 | 0.2812 | 0.5019 |
Entamoeba histolytica | P-glycoprotein-1 | 0.0059 | 1 | 1 |
Trypanosoma cruzi | trans-sialidase, Group I, putative | 0.0031 | 0.2812 | 0.5019 |
Trypanosoma cruzi | trans-sialidase, Group I, putative | 0.0031 | 0.2812 | 0.5019 |
Plasmodium falciparum | multidrug resistance protein 1 | 0.0059 | 1 | 1 |
Trichomonas vaginalis | ABC transporter, putative | 0.0059 | 1 | 1 |
Echinococcus granulosus | ATP binding cassette subfamily B MDR:TAP | 0.0059 | 1 | 1 |
Brugia malayi | P-glycoprotein-like protein | 0.0021 | 0.019 | 0.019 |
Trichomonas vaginalis | ubiquitin-conjugating enzyme E2, putative | 0.0042 | 0.5414 | 0.5414 |
Trichomonas vaginalis | ATP-binding cassette transporter, putative | 0.0059 | 1 | 1 |
Trypanosoma cruzi | ubiquitin-conjugating enzyme E2, putative | 0.0042 | 0.5414 | 1 |
Trypanosoma cruzi | trans-sialidase, Group I, putative | 0.0031 | 0.2812 | 0.5019 |
Echinococcus granulosus | multidrug resistance associated protein 1 | 0.0034 | 0.347 | 0.347 |
Trypanosoma cruzi | ubiquitin-conjugating enzyme E2, putative | 0.0042 | 0.5414 | 1 |
Trypanosoma cruzi | trans-sialidase, putative | 0.0031 | 0.2812 | 0.5019 |
Trypanosoma brucei | trans-sialidase, putative | 0.0031 | 0.2812 | 0.5019 |
Trypanosoma cruzi | multidrug resistance-associated protein, putative | 0.0034 | 0.347 | 0.6278 |
Trichomonas vaginalis | taga, putative | 0.0059 | 1 | 1 |
Mycobacterium ulcerans | component linked with the assembly of cytochrome transport transmembrane ATP-binding protein ABC transporter CydD | 0.0021 | 0.019 | 0.5 |
Trypanosoma brucei | multidrug resistance-associated protein, putative | 0.0034 | 0.347 | 0.6278 |
Brugia malayi | hypothetical protein | 0.0021 | 0.019 | 0.019 |
Loa Loa (eye worm) | ABC transporter transmembrane region family protein | 0.0034 | 0.347 | 0.347 |
Echinococcus multilocularis | ATP binding cassette subfamily B (MDR:TAP) | 0.0059 | 1 | 1 |
Trichomonas vaginalis | ABC transporter, half transporter, putative | 0.0059 | 1 | 1 |
Echinococcus granulosus | ATP binding cassette subfamily B MDR:TAP | 0.0059 | 1 | 1 |
Trichomonas vaginalis | ABC transporter, putative | 0.0059 | 1 | 1 |
Echinococcus granulosus | ATP binding cassette sub family B | 0.0021 | 0.019 | 0.019 |
Trypanosoma cruzi | trans-sialidase, Group I, putative | 0.0031 | 0.2812 | 0.5019 |
Loa Loa (eye worm) | hypothetical protein | 0.0059 | 0.981 | 0.981 |
Schistosoma mansoni | multidrug resistance protein | 0.0021 | 0.019 | 0.019 |
Trypanosoma cruzi | trans-sialidase, Group I, putative | 0.0031 | 0.2812 | 0.5019 |
Giardia lamblia | MRP-like ABC transporter | 0.0034 | 0.347 | 1 |
Chlamydia trachomatis | ABC transporter ATP binding protein/permease | 0.0059 | 1 | 0.5 |
Entamoeba histolytica | P-glycoprotein-5 | 0.0059 | 1 | 1 |
Schistosoma mansoni | ATP-binding cassette sub-family B member 7 mitochondrial precursor (abc7) | 0.0021 | 0.019 | 0.019 |
Trichomonas vaginalis | lipid A export ATP-binding/permease protein msba, putative | 0.0059 | 1 | 1 |
Loa Loa (eye worm) | ubiquitin conjugating enzyme protein 13 | 0.0042 | 0.5414 | 0.5414 |
Echinococcus granulosus | multidrug resistance protein 1 | 0.0059 | 1 | 1 |
Toxoplasma gondii | ABC transporter transmembrane region domain-containing protein | 0.0059 | 1 | 1 |
Trichomonas vaginalis | lipid A export ATP-binding/permease protein msba, putative | 0.0021 | 0.019 | 0.019 |
Loa Loa (eye worm) | ATP-binding cassette sub-family B member 2 | 0.0059 | 1 | 1 |
Entamoeba histolytica | P-glycoprotein 6, putative | 0.0021 | 0.019 | 0.019 |
Echinococcus granulosus | ATP binding cassette sub family B | 0.0021 | 0.019 | 0.019 |
Loa Loa (eye worm) | hypothetical protein | 0.0033 | 0.3279 | 0.3279 |
Leishmania major | p-glycoprotein e | 0.0034 | 0.347 | 0.3343 |
Schistosoma mansoni | smdr1 | 0.0021 | 0.019 | 0.019 |
Echinococcus multilocularis | multidrug resistance associated protein 1 | 0.0034 | 0.347 | 0.3343 |
Toxoplasma gondii | ABC transporter transmembrane region domain-containing protein | 0.0034 | 0.347 | 0.3343 |
Entamoeba histolytica | ubiquitin-conjugating enzyme family protein | 0.0042 | 0.5414 | 0.5414 |
Trichomonas vaginalis | ATP-binding cassette transporter, putative | 0.0059 | 1 | 1 |
Schistosoma mansoni | multidrug resistance protein | 0.0059 | 1 | 1 |
Echinococcus multilocularis | ATP binding cassette subfamily B (MDR:TAP) | 0.0059 | 1 | 1 |
Entamoeba histolytica | hypothetical protein | 0.0034 | 0.347 | 0.347 |
Loa Loa (eye worm) | ABC transporter | 0.0021 | 0.019 | 0.019 |
Echinococcus multilocularis | multidrug resistance protein 1 | 0.0039 | 0.4732 | 0.463 |
Trichomonas vaginalis | ABC transporter, half transporter, putative | 0.0059 | 1 | 1 |
Entamoeba histolytica | ATP-binding cassette protein, putative | 0.0034 | 0.347 | 0.347 |
Echinococcus multilocularis | ubiquitin conjugating enzyme E2 N | 0.0042 | 0.5414 | 0.5325 |
Brugia malayi | ubiquitin conjugating enzyme protein 13 | 0.0042 | 0.5414 | 0.5414 |
Entamoeba histolytica | P-glycoprotein 5, putative | 0.0059 | 1 | 1 |
Echinococcus multilocularis | multidrug resistance protein 1 | 0.0059 | 1 | 1 |
Trypanosoma brucei | p-glycoprotein | 0.0034 | 0.347 | 0.6278 |
Giardia lamblia | ABC transporter, putative | 0.0034 | 0.347 | 1 |
Trichomonas vaginalis | lipid A export ATP-binding/permease protein msba, putative | 0.0059 | 1 | 1 |
Loa Loa (eye worm) | ubiquitin conjugating enzyme protein 13 | 0.0042 | 0.5414 | 0.5414 |
Trichomonas vaginalis | ATP-binding cassette transporter, putative | 0.0059 | 1 | 1 |
Brugia malayi | ABC transporter transmembrane region family protein | 0.0021 | 0.019 | 0.019 |
Plasmodium falciparum | ubiquitin-conjugating enzyme E2 N, putative | 0.0042 | 0.5414 | 0.5325 |
Trichomonas vaginalis | lipid A export ATP-binding/permease protein msba, putative | 0.0059 | 1 | 1 |
Echinococcus multilocularis | ATP binding cassette sub family B | 0.0059 | 0.981 | 0.9806 |
Trichomonas vaginalis | ABC transporter, putative | 0.0059 | 1 | 1 |
Echinococcus multilocularis | multidrug resistance associated protein 7 | 0.0034 | 0.347 | 0.3343 |
Echinococcus granulosus | ubiquitin conjugating enzyme E2 N | 0.0042 | 0.5414 | 0.5414 |
Trypanosoma brucei | trans-sialidase, putative | 0.0031 | 0.2812 | 0.5019 |
Trichomonas vaginalis | lipid A export ATP-binding/permease protein msba, putative | 0.0059 | 1 | 1 |
Trichomonas vaginalis | lipid A export ATP-binding/permease protein msba, putative | 0.0059 | 1 | 1 |
Entamoeba histolytica | ATP-binding cassette protein, putative | 0.0034 | 0.347 | 0.347 |
Trichomonas vaginalis | abcb9, putative | 0.0059 | 1 | 1 |
Mycobacterium ulcerans | transmembrane ABC transporter ATP-binding protein | 0.0021 | 0.019 | 0.5 |
Trichomonas vaginalis | ABC transporter, putative | 0.0059 | 1 | 1 |
Trypanosoma cruzi | trans-sialidase, putative | 0.0031 | 0.2811 | 0.5017 |
Trypanosoma brucei | trans-sialidase, putative | 0.0031 | 0.2812 | 0.5019 |
Entamoeba histolytica | P-glycoprotein 6, putative | 0.0021 | 0.019 | 0.019 |
Trichomonas vaginalis | multidrug resistance protein 1, 2, putative | 0.0059 | 1 | 1 |
Leishmania major | ATP-binding cassette protein subfamily C, member 2, putative | 0.0034 | 0.347 | 0.3343 |
Brugia malayi | multidrug Resistance Protein family member (mrp-5), putative | 0.0021 | 0.019 | 0.019 |
Brugia malayi | ABC transporter | 0.0021 | 0.019 | 0.019 |
Trichomonas vaginalis | multidrug resistance protein 1, 2, putative | 0.0059 | 1 | 1 |
Trichomonas vaginalis | multidrug resistance protein 1, 2, putative | 0.0059 | 1 | 1 |
Trypanosoma cruzi | trans-sialidase, Group I, putative | 0.0031 | 0.2812 | 0.5019 |
Echinococcus multilocularis | ATP binding cassette subfamily B (MDR:TAP) | 0.0059 | 1 | 1 |
Entamoeba histolytica | P-glycoprotein-2 | 0.0059 | 1 | 1 |
Echinococcus granulosus | ATP binding cassette subfamily B MDR:TAP | 0.0059 | 1 | 1 |
Loa Loa (eye worm) | hypothetical protein | 0.0021 | 0.019 | 0.019 |
Trypanosoma cruzi | multidrug resistance-associated protein, putative | 0.0034 | 0.347 | 0.6278 |
Trichomonas vaginalis | lipid A export ATP-binding/permease protein msba, putative | 0.0059 | 1 | 1 |
Trypanosoma cruzi | multidrug resistance protein E, putative | 0.0034 | 0.347 | 0.6278 |
Trypanosoma cruzi | trans-sialidase, Group I, putative | 0.0031 | 0.2812 | 0.5019 |
Entamoeba histolytica | multidrug resistance protein, putative | 0.0034 | 0.347 | 0.347 |
Plasmodium vivax | multidrug resistance protein 1, putative | 0.0059 | 1 | 1 |
Schistosoma mansoni | multidrug resistance protein | 0.0059 | 1 | 1 |
Echinococcus multilocularis | ATP binding cassette subfamily B (MDR:TAP) | 0.0059 | 1 | 1 |
Wolbachia endosymbiont of Brugia malayi | ABC-type multidrug transport system, ATPase and permease component | 0.0021 | 0.019 | 0.5 |
Trypanosoma brucei | multidrug resistance-associated protein, putative | 0.0034 | 0.347 | 0.6278 |
Loa Loa (eye worm) | multidrug resistance protein 3 | 0.0059 | 1 | 1 |
Brugia malayi | ABC transporter family protein | 0.0021 | 0.019 | 0.019 |
Mycobacterium tuberculosis | Probable transmembrane multidrug efflux pump | 0.0059 | 1 | 1 |
Mycobacterium ulcerans | drugs-transport transmembrane ATP-binding protein ABC transporter | 0.0021 | 0.019 | 0.5 |
Leishmania major | ATP-binding cassette protein subfamily C, member 1, putative | 0.0034 | 0.347 | 0.3343 |
Echinococcus granulosus | multidrug resistance protein 1 | 0.0059 | 1 | 1 |
Trichomonas vaginalis | abcb9, putative | 0.0059 | 1 | 1 |
Giardia lamblia | Multidrug resistance-associated protein 1 | 0.0034 | 0.347 | 1 |
Trypanosoma cruzi | trans-sialidase, putative | 0.0031 | 0.2811 | 0.5017 |
Loa Loa (eye worm) | ABC transporter | 0.0021 | 0.019 | 0.019 |
Echinococcus granulosus | multidrug resistance associated protein 7 | 0.0034 | 0.347 | 0.347 |
Schistosoma mansoni | smdr2 | 0.0059 | 1 | 1 |
Wolbachia endosymbiont of Brugia malayi | ABC-type protease secretion system, ATPase and permease component, AprD | 0.0021 | 0.019 | 0.5 |
Schistosoma mansoni | multidrug resistance protein | 0.0034 | 0.347 | 0.347 |
Mycobacterium leprae | PROBABLE DRUGS-TRANSPORT TRANSMEMBRANE ATP-BINDING PROTEIN ABC TRANSPORTER | 0.0021 | 0.019 | 0.5 |
Schistosoma mansoni | ubiquitin conjugating enzyme 13 | 0.0042 | 0.5414 | 0.5414 |
Mycobacterium ulcerans | transmembrane ABC transporter ATP-binding protein | 0.0021 | 0.019 | 0.5 |
Echinococcus multilocularis | multidrug resistance protein 1 | 0.0059 | 1 | 1 |
Giardia lamblia | Multidrug resistance-associated protein 1 | 0.0034 | 0.347 | 1 |
Echinococcus granulosus | multidrug resistance protein 1 | 0.0039 | 0.4732 | 0.4732 |
Leishmania major | ATP-binding cassette protein subfamily C, member 6, putative | 0.0034 | 0.347 | 0.3343 |
Entamoeba histolytica | ABC transporter, putative | 0.0034 | 0.347 | 0.347 |
Trichomonas vaginalis | multidrug resistance protein 1, 2, putative | 0.0059 | 1 | 1 |
Echinococcus granulosus | ATP binding cassette subfamily B MDR:TAP | 0.0059 | 1 | 1 |
Toxoplasma gondii | ATP-binding cassette transporter ABC.B1 | 0.0059 | 1 | 1 |
Brugia malayi | ABC transporter transmembrane region family protein | 0.0034 | 0.347 | 0.347 |
Loa Loa (eye worm) | hypothetical protein | 0.0059 | 1 | 1 |
Loa Loa (eye worm) | hypothetical protein | 0.0034 | 0.347 | 0.347 |
Plasmodium vivax | ubiquitin-conjugating enzyme E2 N, putative | 0.0042 | 0.5414 | 0.5325 |
Mycobacterium ulcerans | transmembrane ABC transporter ATP-binding protein | 0.0021 | 0.019 | 0.5 |
Trichomonas vaginalis | lipid A export ATP-binding/permease protein msba, putative | 0.0059 | 1 | 1 |
Leishmania major | ubiquitin-conjugating enzyme e2, putative | 0.0042 | 0.5414 | 0.5325 |
Trypanosoma cruzi | trans-sialidase, Group I, putative | 0.0031 | 0.2812 | 0.5019 |
Trypanosoma cruzi | trans-sialidase, putative | 0.0031 | 0.2812 | 0.5019 |
Trichomonas vaginalis | ATP-binding cassette transporter, putative | 0.0059 | 1 | 1 |
Leishmania major | ATP-binding cassette protein subfamily B, member 2, putative | 0.0059 | 1 | 1 |
Mycobacterium leprae | PROBABLE DRUGS-TRANSPORT TRANSMEMBRANE ATP-BINDING PROTEIN ABC TRANSPORTER | 0.0021 | 0.019 | 0.5 |
Schistosoma mansoni | multidrug resistance protein | 0.0034 | 0.347 | 0.347 |
Trichomonas vaginalis | multidrug resistance protein 1, 2, putative | 0.0059 | 1 | 1 |
Leishmania major | pentamidine resistance protein 1 | 0.0034 | 0.347 | 0.3343 |
Trypanosoma cruzi | trans-sialidase, putative | 0.0031 | 0.2812 | 0.5019 |
Trypanosoma cruzi | trans-sialidase, putative | 0.0031 | 0.2811 | 0.5017 |
Brugia malayi | ABC transporter family protein | 0.0021 | 0.019 | 0.019 |
Leishmania major | ABC-thiol transporter | 0.0034 | 0.347 | 0.3343 |
Entamoeba histolytica | ATP-binding cassette protein, putative | 0.0034 | 0.347 | 0.347 |
Leishmania major | p-glycoprotein | 0.0059 | 1 | 1 |
Trypanosoma cruzi | trans-sialidase, Group I, putative | 0.0031 | 0.2812 | 0.5019 |
Schistosoma mansoni | multidrug resistance protein | 0.0034 | 0.347 | 0.347 |
Onchocerca volvulus | 0.0059 | 1 | 0.5 | |
Brugia malayi | multidrug resistance related protein 1 | 0.0034 | 0.347 | 0.347 |
Trypanosoma brucei | multidrug resistance protein E | 0.0034 | 0.347 | 0.6278 |
Giardia lamblia | Multidrug resistance-associated protein 1 | 0.0033 | 0.3279 | 0.9452 |
Loa Loa (eye worm) | hypothetical protein | 0.0059 | 1 | 1 |
Trypanosoma brucei | trans-sialidase, putative | 0.0031 | 0.2812 | 0.5019 |
Schistosoma mansoni | multidrug resistance protein | 0.0034 | 0.347 | 0.347 |
Trypanosoma brucei | trans-sialidase, putative | 0.0031 | 0.2812 | 0.5019 |
Trichomonas vaginalis | multidrug resistance protein 1, 2, putative | 0.0059 | 1 | 1 |
Trypanosoma brucei | ubiquitin-protein ligase, putative | 0.0042 | 0.5414 | 1 |
Trichomonas vaginalis | lipid A export ATP-binding/permease protein msba, putative | 0.0059 | 1 | 1 |
Brugia malayi | Ubiquitin conjugating enzyme protein 13 | 0.0042 | 0.5414 | 0.5414 |
Entamoeba histolytica | ATP-binding cassette protein, putative | 0.0034 | 0.347 | 0.347 |
Echinococcus granulosus | 5'partial|ATP binding cassette sub family B | 0.0059 | 0.981 | 0.981 |
Leishmania major | ATP-binding cassette protein subfamily C, member 5, putative | 0.0034 | 0.347 | 0.3343 |
Entamoeba histolytica | P-glyco protein 6, putative | 0.0059 | 1 | 1 |
Echinococcus granulosus | multidrug resistance protein 1 | 0.0059 | 1 | 1 |
Echinococcus multilocularis | ATP binding cassette subfamily B (MDR:TAP) | 0.0059 | 1 | 1 |
Trichomonas vaginalis | ATP-binding cassette transporter, putative | 0.0039 | 0.4732 | 0.4732 |
Brugia malayi | ABC transporter family protein | 0.0021 | 0.019 | 0.019 |
Schistosoma mansoni | multidrug resistance protein | 0.0059 | 1 | 1 |
Trichomonas vaginalis | ATP-binding cassette transporter, putative | 0.0059 | 1 | 1 |
Trichomonas vaginalis | ubiquitin-conjugating enzyme E2, putative | 0.0042 | 0.5414 | 0.5414 |
Activity type | Activity value | Assay description | Source | Reference |
---|---|---|---|---|
Inhibition (functional) | = 44 % | Percent inhibition against ethanol-induced gastric lesions in male albino rat was determined at a dose of 25 mg/Kg | ChEMBL. | 2296028 |
Many chemical entities in TDR Targets come from high-throughput screenings with whole cells or tissue samples, and not all assayed compounds have been tested against a single a single target protein, probably because they get ruled out during screening process. Even if these compounds may have not been of interest in the original screening, they may come as interesting leads for other screening assays. Furthermore, we may be able to propose drug-target associations using chemical similarities and network patterns.
1 literature reference was collected for this gene.